| Cat.No. | Name | Information |
|---|---|---|
| M2347 | (+)-Bicuculline | (+)-Bicuculline is a competitive antagonist of GABAA receptors with IC50 of 2 μM, also blocks Ca(2+)-activated potassium channels. |
| M6319 | 17-PA | 17-PA is a antagonist of neurosteroid potentiation and direct gating of GABA A. |
| M6245 | Basmisanil | Basmisanil is a highly selective GABAAα5 negative allosteric modulator. |
| M6195 | Propofol | Propofol inhibited tumor size, cell viability and promoted cell apoptosis via inhibiting mTOR/p70S6K pathway mediated by HOTAIR in cervical cancer. |
| M6010 | Tiagabine HCl | Tiagabine Hydrochloride is the hydrochloride salt form of tiagabine, a nipecotic acid derivative with anticonvulsant property. A selective gamma-aminobutyric acid (GABA) reuptake inhibitor. |
| M6009 | Tiagabine | Tiagabine is an anticonvulsant compound that acts as an inhibitor of GABA reabsorption. |
| M5870 | Pentylenetetrazol | Pentylenetetrazol displays activity as a central nervous system and respiratory stimulant. It is considered a non-competitive GABA(A) receptor antagonist. |
| M5730 | L-Cycloserine | L-cycloserine irreversibly inhibit GABA pyridoxal 5′-phosphate-dependent aminitransferase in E. coli, as well in the brains of various animals in a time-dependent manner, results in increased levels of gamma-aminobutyric acid (GABA), which is an inhibitory neurotransmitter in vivo. |
| M5669 | Gabapentin HCl | Gabapentin HCl is a GABA analogue, used to treat seizures and neuropathic pain. |
| M5653 | Flumazenil | Flumazenil is a competitive GABAA receptor antagonist, used in the treatment of benzodiazepine overdoses. |
| M5575 | Dihydroergotoxine mesylate | Dihydroergotoxine mesylate is a complex of closely related alkaloid salts; Binds with high affinity to the GABAA receptor Cl- channel, producing an allosteric interaction with the benzodiazepine site. |
| M5442 | Baclofen | Baclofen is a gamma-amino-butyric acid (GABA) derivative used as a skeletal muscle relaxant. |
| M5390 | Afloqualone | Afloqualone is a agonist of GABA receptor . |
| M5378 | Acamprosate calcium | Acamprosate calcium (Campral EC) is a GABA receptor agonist and glutamate system modulator. |
| M4959 | Pagoclone | Pagoclone, active (+)-enantiomer of the racemate RP 59037, is a partial GABA(A) receptor agonist that used for treatment of panic and anxiety disorders. |
| M4815 | Vigabatrin | Vigabatrin (γ-Vinyl-GABA), an inhibitory neurotransmitter GABA vinyl-derivative, is an orally active and irreversible GABA transaminase inhibitor. |
| M4441 | Jujuboside-A | Jujuboside A is A glycoside extracted from the Chinese traditional medicine ziziphus jujuboides, which can be used in studies on insomnia and anxiety symptoms. |
| M4231 | Ginkgolide-A | Ginkgolide A (BN-52020) is A GABA antagonist extracted from ginkgo biloba leaves. |
| M4073 | Ginsenoside-Rc | Ginsenoside Rc is one of the major ginsenosides. Ginsenoside Rc enhances GABA receptor A (GABAA) -mediated ion channel (IGABA) currents. Ginsenoside Rc also inhibited TNF-α and IL-1β expression. |
| M4019 | Songorine | Songorine is a diterpenoid alkaloid isolated from the genus Aconite. Songorine is a GABAA receptor antagonist in rat brain and has anticancer, anti-arrhythmia and anti-inflammatory activities. Songorine has potential to be used in epithelial ovarian cancer (EOC) studies. |
| M4013 | Glabridin | Glabridin, one of the active phytochemicals in licorice extract, binds to and activates the ligand binding domain of PPARγ, as well as the full length receptor. It is also a GABAA receptor positive modulator promoting fatty acid oxidation and improving learning and memory. |
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