| Cat.No. | Name | Information |
|---|---|---|
| M2347 | (+)-Bicuculline | (+)-Bicuculline is a competitive antagonist of GABAA receptors with IC50 of 2 μM, also blocks Ca(2+)-activated potassium channels. |
| M10326 | Zuranolone | Zuranolone also known as SAGE-217, is a potent GABAA receptor agonist with EC50 values of 296 nM and 163 nM for α1β2γ2 and α4β3δ GABAA receptors. |
| M9874 | SSD114 hydrochloride | SSD114 hydrochloride is a GABAB receptor positive allosteric modulator. |
| M9856 | Pipequaline | Pipequaline (PK-8165) is a partial benzodiazepine receptor agonist with anxiolytic activity. |
| M9411 | AZD-7325 | AZD-7325 is a GABA-Aα2,3 -selective receptor modulator. |
| M9188 | Clomethiazole | Clomethiazole is a positive allosteric modulator at the barbiturate/picrotoxin site of the GABAA receptor. |
| M9127 | ONO-8590580 | ONO-8590580 is a GABAAα5 negative allosteric modulator which enhances long-term potentiation and improves cognitive deficits in preclinical models. |
| M9114 | LAU159 | LAU159 is a potent, functionally selective α6β3γ2 GABAA receptor modulator. |
| M8879 | Aminooxy-acetic acid (AOA) hemihydrochloride | Aminooxyacetic acid hemihydrochloride is a malate-aspartate shuttle (MAS) inhibitor which also inhibits the GABA degradating enzyme GABA-T. |
| M8216 | Securinine | Securinine is an alkaloid widely in traditional folk medicine, it is a GABAA receptor antagonist. |
| M8027 | 5α-Pregnan-3α-ol-20-one | Positive allosteric modulator of GABAA chloride channel. |
| M7813 | Isoguvacine hydrochloride | Isoguvacine hydrochloride is a GABAA receptor agonist. |
| M7691 | Chlormethiazole hydrochloride | Chlormethiazole hydrochloride is a GABAA agonist; glycine receptor modulator. |
| M7607 | 5α-Androst-16-en-3α-ol | 5alpha-androst-16-en-3alp |
| M7442 | U 93631 | U 93631 is a gABA A receptor antagonist. |
| M7410 | THIP hydrochloride | THIP hydrochloride is a gABA A agonist. |
| M7252 | SB 205384 | SB 205384 is a gABA A receptor modulator; slows current decay. |
| M7242 | Saclofen | Saclofen is a selective GABA B antagonist. |
| M6744 | Ganaxolone | Ganaxolone (CCD 1042) is A neuroactive steroid allopregnenolone analogue synthesized orally and is A selective, high-affinity positive sex modulator of γ -aminobutyrate-A (GABAA) receptor with anticonvulsant properties. Gannadone works through different binding sites with benzodiazepine binding sites and can be used in epilepsy studies related to cyclin-dependent kinase-like 5 (CDKL5) deficiency (CDD). |
| M6720 | Etifoxine hydrochloride | Etifoxine hydrochloride is a ligand of the translocator protein (TSPO); also GABA A receptor potentiator. |
| M6585 | CGP52432 | CGP 52432 is a potent, selective GABAB antagonist. |
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