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THIP (Gaboxadol) is a selective δ-aminobutyric acid type A receptor (δ-GABAAR) agonist, functionally selective GABAAR ligand, exhibits agonism at α4β1δ, α4β3δ and weak antagonism at αβγ and α4β2δ GABAARs.
| Molecular Weight | 140.14 |
| CAS Number | 64603-91-4 |
| Solubility (25°C) | DMSO 90 mg/mL (ultrasonic and adjust pH to 3 with HCl) Water 23.33 mg/mL |
| Storage |
Powder -20°C 3 years ; 4°C 2 years In solvent -80°C 6 months ; -20°C 1 month |
[1] W Wisden, et al. GABA Receptors and the Pharmacology of Sleep
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