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GABA Receptor GABA Receptor

Inhibitors

Cat.No.  Name Information
M10326 Zuranolone Zuranolone also known as SAGE-217, is a potent GABAA receptor agonist with EC50 values of 296 nM and 163 nM for α1β2γ2 and α4β3δ GABAA receptors.
M9874 SSD114 hydrochloride SSD114 hydrochloride is a GABAB receptor positive allosteric modulator.
M9856 Pipequaline Pipequaline (PK-8165) is a partial benzodiazepine receptor agonist with anxiolytic activity.
M9411 AZD-7325 AZD-7325 is a GABA-Aα2,3 -selective receptor modulator.
M9127 ONO-8590580 ONO-8590580 is a GABAAα5 negative allosteric modulator which enhances long-term potentiation and improves cognitive deficits in preclinical models.
M9114 LAU159 LAU159 is a potent, functionally selective α6β3γ2 GABAA receptor modulator.
M8879 AOA hemihydrochloride Aminooxyacetic acid hemihydrochloride is a malate-aspartate shuttle (MAS) inhibitor which also inhibits the GABA degradating enzyme GABA-T.
M8027 5α-Pregnan-3α-ol-20-one Positive allosteric modulator of GABAA chloride channel.
M7691 Chlormethiazole hydrochloride Chlormethiazole hydrochloride is a GABAA agonist; glycine receptor modulator.
M6744 Ganaxolone Ganaxolone (CCD 1042) is A neuroactive steroid allopregnenolone analogue synthesized orally and is A selective, high-affinity positive sex modulator of γ -aminobutyrate-A (GABAA) receptor with anticonvulsant properties. Gannadone works through different binding sites with benzodiazepine binding sites and can be used in epilepsy studies related to cyclin-dependent kinase-like 5 (CDKL5) deficiency (CDD).
M6585 CGP52432 CGP 52432 is a potent, selective GABAB antagonist.
M6195 Propofol Propofol inhibited tumor size, cell viability and promoted cell apoptosis via inhibiting mTOR/p70S6K pathway mediated by HOTAIR in cervical cancer.
M6010 Tiagabine HCl Tiagabine Hydrochloride is the hydrochloride salt form of tiagabine, a nipecotic acid derivative with anticonvulsant property. A selective gamma-aminobutyric acid (GABA) reuptake inhibitor.
M6009 Tiagabine Tiagabine is an anticonvulsant compound that acts as an inhibitor of GABA reabsorption.
M5870 Pentylenetetrazol Pentylenetetrazol displays activity as a central nervous system and respiratory stimulant. It is considered a non-competitive GABA(A) receptor antagonist.
M5730 L-Cycloserine L-cycloserine irreversibly inhibit GABA pyridoxal 5′-phosphate-dependent aminitransferase in E. coli, as well in the brains of various animals in a time-dependent manner, results in increased levels of gamma-aminobutyric acid (GABA), which is an inhibitory neurotransmitter in vivo.
M5669 Gabapentin HCl Gabapentin HCl is a GABA analogue, used to treat seizures and neuropathic pain.
M5653 Flumazenil Flumazenil is a competitive GABAA receptor antagonist, used in the treatment of benzodiazepine overdoses.
M5575 Dihydroergotoxine mesylate Dihydroergotoxine mesylate is a complex of closely related alkaloid salts; Binds with high affinity to the GABAA receptor Cl- channel, producing an allosteric interaction with the benzodiazepine site.
M5442 Baclofen Baclofen is a gamma-amino-butyric acid (GABA) derivative used as a skeletal muscle relaxant.



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