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CNS 7056 is a short-acting GABAa receptor agonist used in general anesthesia.
| Molecular Weight | 439.31 |
| Formula | C21H19BrN4O2 |
| CAS Number | 308242-62-8 |
| Storage | 2-8℃ |
[2] J Robert Sneyd, et al. Curr Opin Anaesthesiol. Remimazolam for anaesthesia or sedation
| Related GABA Receptor Products |
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| TPMPA
TPMPA, a hybrid of isoguvacine and 3-APMPA, is the first selective antagonist for a GABAC receptor (KB = 2.1 μM), but not to interact with GABAA (KB = 320 μM) or GABAB receptors (EC50 = 500 μM). |
| CI-966
CI-966 is a potent, selective, orally active and brain-penetrant inhibitor of the GABA transporter GAT-1, with IC50s of 0.26 μM and 1.2 μM for hGAT-1, rGAT-1, respectively. |
| NCS-382
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| CGS 8216
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