| Cat.No. | Name | Information |
|---|---|---|
| M2347 | (+)-Bicuculline | (+)-Bicuculline is a competitive antagonist of GABAA receptors with IC50 of 2 μM, also blocks Ca(2+)-activated potassium channels. |
| M42188 | Xilmenolone | Xilmenolone is a GABAA receptor positive allosteric modulator. |
| M42187 | NNC 05-2090 | NNC 05-2090 is a potent inhibitor of mGAT2, with a Ki of 1.4 μM. |
| M42186 | Arecaidine hydrobromide | Arecaidine hydrobromide, a pyridine alkaloid, is a potent GABA uptake inhibitor. |
| M42185 | Muscimol hydrochloride | Muscimol (Agarin; Agarine) hydrochloride is an isoxazole with psychoactive activity. |
| M42184 | γ-Acetylenic GABA hydrochloride | γ-Acetylenic GABA (GAG) hydrochloride is an irreversible inhibitor of GABA-transaminase. |
| M42183 | Panadiplon | Panadiplon (FG 10571; PNU 78875), a benzodiazepine receptor, is a 5GABAA partial agonist. |
| M42182 | α5IA | α5IA (L-822179) is a selective α5 GABAA receptor inverse agonist with neuroprotective potential. |
| M42181 | 3-Methylglutaconic acid | 3-Methylglutaconic acid is the major metabolites accumulating in 3-Methylglutaconic aciduria (MGTA). |
| M42180 | Guvacine hydrobromide | Guvacine hydrobromide, an alkaloid found in the nut of Areca catechu, is a potent GABA uptakp inhibitor. |
| M42179 | CGS 20625 | CGS 20625 is a potent, selective and orally active partial agonist for the central benzodiazepine receptor. |
| M42178 | 1-Phenyl-2-pyrrolidinone | 1-Phenyl-2-pyrrolidinone (1-Phenylpyrrolidin-2-one) is a phenyl analogue of GABA with sedative effect, decreasing the exploratory behavior of rats at 50-100 mg/kg (i.v.). |
| M42177 | SCS | SCS (Salicylidene salicylhydrazide) is a potent, allosteric and selective inhibitor of β1-containing GABAA receptors with an IC50 of 32 nM against α2β1γ1θ by VIPR measurement. |
| M39028 | Picrotin | Picrotin is an active compound, also is one of the composition of picrotoxin (an antagonist of GABAA receptors (GABAARs) and glycine receptors (GlyRs)). Picrotin has sensitivity for GlyRs/b> with IC50 values range from 5.2 μM to 106 μM. Picrotin can be used for the research of neurotransmission. |
| M39027 | Isohyenanchin | Isohyenanchin (Hydroxycoriatin) is an RDLac homo-oligomers antagonist. Isohyenanchin also is a weak antagonist of ionotropic GABA receptors. |
| M39026 | Chrodrimanin B | Chrodrimanin B is a potent, non-open-channel-blocking antagonist on B. mori GABAR RDL with an IC50 of 1.13 nM. Chrodrimanin B attenuates the peak current amplitude of the GABA response of RDL with an IC50 of 1.66 nM. |
| M39025 | Isonipecotic acid | Isonipecotic acid is a GABAA receptor partial agonist. |
| M39024 | Guvacine ethyl ester | Guvacine ethyl ester (3.1b) is an alkaloid that can be found in betel nut. Guvacine ethyl ester can be used in the synthesis of GABA uptake inhibitor. |
| M39023 | 6-Aminonicotinic acid | 6-Aminonicotinic acid is a GABAA receptor agonist with Ki value of 4.4 nM. |
| M39022 | 3,4,5-Trimethoxycinnamic acid | 3,4,5-Trimethoxycinnamic acid has anti-stress effect, prolonging the sleeping time in animals. 3,4,5-Trimethoxycinnamic acid increases expression of GAD65 and γ-subunit of GABAA receptor, but shows no effect on the amounts of α-, β-subunits. |
| M31352 | Progabide | Progabide is a gamma-aminobutyric acid (GABA) receptor agonist that may be used in studies related to epilepsy. |
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