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Clomethacazole is a thiol (vitamin B1)-related compound that acts as a thiazole derivative. Clomethiazole is a positive allosteric modulator at the barbiturate/picrotoxin site of the GABAA receptor. It acts as a sedative and hypnotic agent.
| Molecular Weight | 161.64 |
| Formula | C6H8ClNS |
| CAS Number | 533-45-9 |
| Solubility (25°C) | DMSO 10 mM |
| Storage | 4°C, dry, sealed |
[2] No authors listed. Drugs R D. Clomethiazole. Chlormethiazole, Zendra
[4] E Klug, et al. Clomethiazole poisoning
[5] P Lechat. Toxicological and pharmacological properties of clomethiazole
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