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Chlormethiazole hydrochloride is a GABAA agonist; glycine receptor modulator. Clomethiazole hydrochloride is neuroprotective and prevents the degeneration of serotonergic nerve terminals induced by 3,4-methylenedioxymethamphetamine (MDMA).
| Molecular Weight | 198.11 |
| Formula | C6H8ClNS.HCl |
| CAS Number | 6001-74-7 |
| Solubility (25°C) | Water 90 mg/mL DMSO 100 mg/mL |
| Storage |
Powder -20°C 3 years ; 4°C 2 years In solvent -80°C 6 months ; -20°C 1 month |
[4] S K Majumdar. Chlormethiazole and utilization of vitamin B1 in chronic alcoholics
[5] No authors listed. Drug Intell Clin Pharm. Drug interactions with medical plastics
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