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Acamprosate calcium

Cat. No. M5378

All AbMole products are for research use only, cannot be used for human consumption.

Acamprosate calcium Structure
Synonym:

Calcium N-acetylhomotaurinate

Size Price Availability Quantity
50mg USD 60  USD60 In stock
250mg USD 180  USD180 In stock
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Quality Control & Documentation
Biological Activity

Acamprosate, or N-acetyl homotaurine, is an N-methyl-D-aspartate receptor modulator approved by the Food and Drug Administration (FDA) as a pharmacological treatment for alcohol dependence.Acamprosate has low bioavailability, but also has an excellent tolerability and safety profile. In comparison with naltrexone and disulfiram, which are the other FDA-approved treatments for alcohol dependence, acamprosate is unique in that it is not metabolized by the liver and is also not impacted by alcohol use, so can be administered to patients with hepatitis or liver disease (a common comorbid condition among individuals with alcohol dependence) and to patients who continue drinking alcohol.

Chemical Information
Molecular Weight 200.24
Formula 2(C5H10NO4S).Ca
CAS Number 77337-73-6
Form Solid
Solubility (25°C) H2O 90 mg/mL
Storage 4°C, dry, sealed
References

[1] Spanagel R, et al. Neuropsychopharmacology. Acamprosate produces its anti-relapse effects via calcium.

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Keywords: Acamprosate calcium, Calcium N-acetylhomotaurinate supplier, GABA Receptor, inhibitors, activators

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