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SB 205384 is a gABAA receptor modulator; slows current decay. Potentiates α6, α3 and α5-subunit-containing receptors (EC50 values are 280, 695 and 730 nM respectively). Displays little effect on receptors containing α1 or α2 subunits.
| Molecular Weight | 330.4 |
| Formula | C17H18N2O3S |
| CAS Number | 160296-13-9 |
| Solubility (25°C) | 1eq. HCl 33.04 mg/mL |
| Storage |
Powder -20°C 3 years ; 4°C 2 years In solvent -80°C 6 months ; -20°C 1 month |
| Related GABA Receptor Products |
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| TPMPA
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| CGS 8216
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