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Ganaxolone

Cat. No. M6744

All AbMole products are for research use only, cannot be used for human consumption.

Ganaxolone Structure
Synonym:

CCD 1042

Size Price Availability Quantity
5mg USD 200  USD200 In stock
10mg USD 285  USD285 In stock
25mg USD 510  USD510 In stock
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Quality Control & Documentation
Biological Activity

Ganaxolone (CCD 1042) is A neuroactive steroid allopregnenolone analogue synthesized orally and is A selective, high-affinity positive sex modulator of γ -aminobutyrate-A (GABAA) receptor with anticonvulsant properties. Gannadone works through different binding sites with benzodiazepine binding sites and can be used in epilepsy studies related to cyclin-dependent kinase-like 5 (CDKL5) deficiency (CDD).

Chemical Information
Molecular Weight 332.53
Formula C22H36O2
CAS Number 38398-32-2
Solubility (25°C) DMSO 3.33 mg/mL (with gentle warming)
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Castanho, et al. J Biol Chem. Absorption and fluorescence spectra of polyene antibiotics in the presence of cholesterol.

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Keywords: Ganaxolone, CCD 1042 supplier, GABA Receptor, inhibitors, activators

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