Cat.No. | Name | Information |
---|---|---|
M2489 | Carbachol chloride | Carbachol is a cholinomimetic compound that binds and activates the acetylcholine receptor. |
M3470 | Oxybutynin | Oxybutynin is an anticholinergic medication used to relieve urinary and bladder difficulties. |
M3190 | PNU-282987 | PNU-282987 is a highly selective α7 nAChR agonist with Ki of 27 nM. |
M5683 | Glycopyrrolate | Glycopyrrolate(Glycopyrronium Br) is a muscarinic competitive antagonist used as an antispasmodic. |
M3601 | Donepezil hydrochloride | Donepezil is a specific and potent AChE inhibitor for bAChE and hAChE with IC50 of 8.12 nM and 11.6 nM , respectively. |
M3590 | Butylscopolamine Bromide | Butylscopolamine Bromide, is a peripherally acting antimuscarinic, anticholinergic agent used as an abdominal-specific antispasmodic. |
M3589 | Methscopolamine bromide | Methscopolamine is a muscarinic acetylcholine receptor blocker. |
M3534 | Pancuronium dibromide | Pancuronium dibromide is a competitive acetylcholine antagonist with an IC50 of 5.5 nM. |
M3530 | Tolterodine tartrate | Tolterodine tartrate is a tartrate salt of tolterodine that is a competitive muscarinic receptor antagonist. |
M3501 | Ipratropium Bromide | Ipratropium Bromide is a muscarinic antagonist, bronchodilator, N-Isopropyl salt of atropine. |
M3403 | PNU-120596 | PNU-120596 is a positive allosteric modulator of α7 nAChR with EC50 of 216 nM. |
M3401 | 5-hydroxymethyl Tolterodine | 5-hydroxymethyl tolterodine (PNU 200577) is a new muscarinic receptor antagonist with Kb of 0.84 nM. |
M3393 | Pyridostigmine Bromide | Pyridostigmine Bromide is a parasympathomimetic and a reversible cholinesterase inhibitor. |
M3331 | Trospium chloride | Trospium chloride is an orally active, competitive muscarinic cholinergic receptors (mAChRs) antagonist. Trospium chloride binds to muscarinic receptors M1, M2 and M3 with high affinity, but not nicotinic, cholinergic receptors. |
M3317 | Acetylcholine Chloride | The chemical compound Acetylcholine Chloride is a neurotransmitter in both the peripheral nervous system (PNS) and central nervous system (CNS) in many organisms including humans. |
M3309 | Bethanechol chloride | Bethanechol chloride is a selective muscarinic receptor agonist without any effect on nicotinic receptors. Bethanechol chloride (0.3-300 μM) significantly reduces ileal pacemaker potentials. |
M3253 | (-)-Huperzine A | (-)-Huperzine A is a potent, highly specific and reversible inhibitor of acetylcholinesterase (AChE) with Ki of 7 nM, exhibiting 200-fold more selectivity for G4 AChE over G1 AChE. Also acts as an NMDA receptor antagonist. Phase 4. |
M3225 | Atropine sulfate | Atropine sulfate is a competitive muscarinic acetylcholine receptor antagonist. |
M3046 | Tacrine hydrochloride | Tacrine is a centrally acting anticholinesterase and indirect cholinergic agonist. |
M3034 | Succinylcholine Chloride Dihydrate | Succinylcholine Chloride Dihydrate is a nicotinic AChR agonist and also acts as a depolarizing neuromuscular blocker. |
M3025 | Solifenacin succinate | Solifenacin succinate is an anti-muscarinic urinary spasmolysis compound. Solifenacin Succinate (YM905) is a novel muscarinic receptor antagonist with pKis of 7.6, 6.9 and 8.0 for M1, M2 and M3 receptors, respectively. |
M2957 | Pridinol Methanesulfonate | Pridenol mesylate is used as an anticholinergic compound and an antiparkinsonian compound. |
M2947 | Pipenzolate Bromide | Pipenzolate is an antimuscarinic, which binds to muscarinic receptors as an antagonist therefore preventing acetyl choline from binding to the receptors. |
M2939 | Physostigmine Salicylate | Physostigmine is a parasympathomimetic alkaloid, specifically, a reversible cholinesterase inhibitor. |
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