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Opioid Receptor Opioid Receptor

Cat.No.  Name Information
M4808 TRV130 hydrochloride TRV130 (Oliceridine) hydrochloride is a novel μ-opioid receptor (MOR) G protein-biased ligand.
M1579 Naloxone Naloxone is an opioid inverse agonist drug used to counter the effects of opiate overdose.
M9615 DAMGO DAMGO is an opioid receptor agonist with the ability to affect the locomotive activity in rodents, Kd value is 3.46 nM for native μ-OPR.
M10432 Difelikefalin (CR-845; FE-202845) TFA Difelikefalin (CR-845; FE-202845) TFA is a synthetic peptide and the first-in-class, peripherally-restricted, selective agonist of the κ-opioid receptor (KOR) for studies related to pruritus.
M10240 CTOP TFA CTOP TFA is a peptide that acts as a potent and selective μ opioid receptor antagonist, with Ki values of 0.96 and >10,000 nM for μ and δ receptors, respectively.
M10229 Porcine dynorphin A (1-13) Porcine dynorphin A (1-13) is a potent, endogenous κ opioid receptor agonist.
M9784 Naloxegol oxalate Naloxegol oxalate (NKTR-118 oxalate; AZ-13337019 oxalate) is a peripherally-selective opioid antagonist for the treatment of opioid-induced constipation.
M9514 JDTic JDTic is a kappa opioid receptor (KOR) antagonist that prevents stress-induced reinstatement of cocaine-maintained responding and has antidepressant-like effects.
M9268 Met-Enkephalin Met-Enkephalin (H-Tyr-Gly-Gly-Phe-Met-OH) inhibits tumor growth via binding to the opioid receptor.
M8502 Alvimopan Alvimopan is a gastroprokinetic peripheral mu-opioid receptor antagonist.
M6036 Trimebutine maleate Trimebutine maleate is a drug with antimuscarinic and weak mu opioid agonist effects.
M6035 Trimebutine Trimebutine is an agonist of peripheral mu, kappa and delta opiate receptors, used as spasmolytic agent for treatment of both acute and chronic abdominal pain.
M5589 Docusate Sodium Docusate Sodium is a compound used to study constipation.
M5403 Alvimopan dihydrate Alvimopan dihydrate (ADL 8-2698 dihydrate) is a potent, selective, orally active and reversible μ-opioid receptor antagonist, with an IC50 of 1.7 nM. Alvimopan dihydrate has selectivity for μ-opioid receptor (Ki=0.47 nM) over κ- and δ-opioid receptors (Kis=100, 12 nM, respectively).
M5289 PZM21 PZM21 is a potent and selective μ-opioid-receptor (μOR) agonist with an EC50 of 1.8 nM.
M5067 Eluxadoline Eluxadoline is an orally active mixed μ opioid receptor (μOR) agonist δ opioid receptor (δOR) antagonist.
M5065 Cebranopadol Cebranopadol is a NOP and opioid receptor agonist that acts on human NOP, MOP, KOP and δ-opioid peptide (DOP) receptors with Ki/EC50 values of 0.9 nM/13 nM and 0.7 nM/1.2 nM, respectively. 2.6 nM/17 nM, 18 nM/110 nM.
M4456 Sec-O-Glucosylhamaudol Sec-o-glucosylhamaudol is a natural product isolated from The apostrophophore, which can reduce the protein level of μ-opioid receptor and can be used for pain relief research.
M3240 MCOPPB trihydrochloride MCOPPB trihydrochloride is a trihydrochloride form of MCOPPB that is a new nonpeptide nociceptin/orphanin FQ peptide (NOP)-receptor agonist with a pKi of 10.07 ±0.01 for the human NOP recepto
M2876 Naloxone hydrochloride Naloxone hydrochloride is an opioid inverse agonist compound used to counter the effects of opiate overdose.
M2875 Nalmefene hydrochloride Nalmefene is an opioid receptor antagonist, it is used primarily in the management of alcohol dependence.
M2838 Meptazinol hydrochloride Meptazinol is a unique centrally active opioid analgesic, which inhibits [3H]dihydromorphine binding with IC50 of 58 nM.
M2214 JTC-801 JTC-801 is a novel opioid receptor-like1 (ORL1) receptor antagonist with IC50 of 94 nM.




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