| Cat.No. | Name | Information |
|---|---|---|
| M4808 | TRV130 hydrochloride | TRV130 (Oliceridine) hydrochloride is a novel μ-opioid receptor (MOR) G protein-biased ligand. |
| M1579 | Naloxone | Naloxone is an opioid inverse agonist drug used to counter the effects of opiate overdose. |
| M9615 | DAMGO | DAMGO is an opioid receptor agonist with the ability to affect the locomotive activity in rodents, Kd value is 3.46 nM for native μ-OPR. |
| M2876 | Naloxone hydrochloride | Naloxone hydrochloride is an opioid inverse agonist compound used to counter the effects of opiate overdose. |
| M2875 | Nalmefene hydrochloride | Nalmefene is an opioid receptor antagonist, it is used primarily in the management of alcohol dependence. |
| M2838 | Meptazinol hydrochloride | Meptazinol is a unique centrally active opioid analgesic, which inhibits [3H]dihydromorphine binding with IC50 of 58 nM. |
| M2214 | JTC-801 | JTC-801 is a novel opioid receptor-like1 (ORL1) receptor antagonist with IC50 of 94 nM. |
| M1953 | ADL5859 Hydrochloride | ADL5859 is a potent, selective and orally bioavailable δ-opioid receptor agonist (Ki = 0.84 nM, EC50 = 20 nM). |
| M1585 | 6-Alpha Naloxol | 6-Alpha Naloxol |
| M1577 | Naltrexone Hydrochloride | Naltrexone hydrochlorideis an opioid receptor antagonist used primarily in the management of alcohol dependence and opioid dependence. |
| M56298 | SNC162 | SNC162 is a delta-opioid receptor agonist with an IC50 of 0.94 nM. |
| M56297 | ML 190 | ML 190 is a selective κ opioid receptor (KOR) antagonist with an IC50 of 120 nM and an EC50 of 129 nM, respectively. |
| M56296 | CCG258747 | CCG258747 is a selective GRK2 inhibitor (IC50=18 nM) with high selectivity over GRK1, GRK5, PKA, and ROCK1 (518, 83, >5500, and >550–fold, respectively).CCG258747 also blocks the internalization of the µ-opioid receptor. |
| M56295 | Sunobinop | Sunobinop (S 117957) is a modulator of the opioid receptor-like orphan receptor (ORL1). |
| M56294 | SCH 486757 | SCH 486757 is an orally effective pain peptide receptor (NOP) agonist. |
| M56293 | Ac-RYYRWK-NH2 | Ac-RYYRWK-NH2 is a potent and selective partial agonist for the nociceptin receptor (NOP), [3H]Ac-RYYRWK-NH2 binds to rat cortical membranes ORL1 with a Kd of 0.071 nM, but has no affinity for µ-, κ- or δ-opioid receptors. |
| M56292 | Ac-RYYRWK-NH2 TFA | Ac-RYYRWK-NH2 is a potent and selective partial agonist for the nociceptin receptor (NOP), [3H]Ac-RYYRWK-NH2 binds to rat cortical membranes ORL1 with a Kd of 0.071 nM, but has no affinity for μ-, κ- or δ-opioid receptors. |
| M56291 | LY2940094 tartrate | LY2940094 (BTRX-246040) tartrate is a potent, brain penetrant, selective and orally available N/OFQ peptide (NOP) receptor antagonist with high affinity (Ki=0.105 nM) and antagonist potency (Kb=0.166 nM). |
| M56290 | AR-M 1000390 hydrochloride | AR-M 1000390 hydrochloride is an exceptionally selective, potent δ opioid receptor agonist with an EC50 of 7.2±0.9 nM for δ agonist potency. |
| M56289 | (-)-U-50488 hydrochloride | (-)-U-50488 hydrochloride ((-)-Trans-(1S,2S)-U-50488 hydrochloride) is a selective kappa-opioid receptor (KOR) agonist (b>Kd=2.2 nM) over μ-opioid receptor (MOR) (b>Kd=430 nM). |
| M54828 | Tegileridine | Tegileridine is the potent agonist of opioid receptor (MOR). Tegileridine is an oxa spiro derivative which reduces the side effects mediated by β-arrestin. |
| M54435 | Morphiceptin | Morphiceptin is a potent and specific agonist for morphine (μ) receptors. |
| M54425 | [Met5]-Enkephalin, amide TFA | [Met5]-Enkephalin, amide TFA is an agonist for δ opioid receptors as well as putative ζ (zeta) opioid receptors. |
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