| Cat.No. | Name | Information |
|---|---|---|
| M4808 | TRV130 hydrochloride | TRV130 (Oliceridine) hydrochloride is a novel μ-opioid receptor (MOR) G protein-biased ligand. |
| M1579 | Naloxone | Naloxone is an opioid inverse agonist drug used to counter the effects of opiate overdose. |
| M9615 | DAMGO | DAMGO is an opioid receptor agonist with the ability to affect the locomotive activity in rodents, Kd value is 3.46 nM for native μ-OPR. |
| M52978 | [Nphe1]Nociceptin(1-13)NH2 | [Nphe1]Nociceptin(1-13)NH2, a novel nociceptin/orphanin FQ (NC) endogenous ligand, is a selective and competitive ociceptin receptor antagonist without any residual agonist activity. |
| M52977 | [Arg14, Lys15]Nociceptin | [Arg14,Lys15]Nociceptin is a highly potent and selective NOP receptor (ORL1; OP4) agonist, with an EC50 of 1 nM. |
| M52976 | D-Ala-Gly-Phe-Met-NH2 monoacetate | D-Ala-Gly-Phe-Met-NH2 monoacetate, an opioid peptide, is a potent opiate δ-receptor agonist. |
| M52975 | β-Endorphin (1-27) (human) | β-Endorphin (1-27) (human) is an opioid antagonist that binds μ-, δ-, and κ-opioid receptors with Kis of 5.31, 6.17, and 39.82 nM, respectively. |
| M52974 | β-Endorphin (6-31), human | β-Endorphin, an endogenous opioid neuropeptide, is an opioid receptor agonist. |
| M52973 | 2, 6-Dimethyl-L-tyrosine | 2,6-Dimethyl-L-tyrosine (Dmt) is a tyrosine derivative that enhances receptor affinity, functional bioactivity and in vivo analgesia of opioid peptides. |
| M52972 | Nociceptin (1-13), amide | Nociceptin (1-13), amide is a potent ORL1 receptor (opioid receptor-like 1 receptor, OP4) agonist with a pEC50 of 7.9 for mouse vas deferens and a Ki of 0.75 nM for binding to rat forebrain membranes. |
| M52971 | Neuropeptide AF (human) | Neuropeptide AF (human) is an endogenous antiopioid peptide. |
| M52970 | D-Ala-Gly-Phe-Met-NH2 | D-Ala-Gly-Phe-Met-NH2, an opioid peptide, is a potent opiate δ-receptor agonist. |
| M52969 | β-Casomorphin, human | is an opioid peptide, acts as an agonist of opioid receptor. |
| M52968 | β-Lipotropin (60-65) | β-Lipotropin (60-65) (β-LPH (60-65)), an opioid peptide, is a potent opioid agonist. |
| M52967 | Dynorphin B (1-9) | Dynorphin B (1-9) is a neuropeptide and N-terminal cleavage product of dynorphin B. |
| M52966 | Leumorphin, human | Leumorphin, human is a potent kappa opioid receptor (κ opioid receptor) agonist. |
| M52965 | Orphanin FQ(1-11) | Orphanin FQ(1-11), a orphanin FQ or nociceptin (OFQ/N) fragment, is a potent NOP receptor (ORL-1; OP4) agonist, with a Ki of 55 nM. |
| M52964 | β-Endorphin (rat) | β-Endorphin (rat) is an endogenous opioid neuropeptide and peptide hormone. |
| M52963 | Helianorphin-19 | Helianorphin-19 is a potent and selective κ-opioid receptor (KOR) activator with a Ki of 21 nM and an EC50 of 45 nM. |
| M52962 | Nociceptin(1-7) | Nociceptin (1-7) is the N-terminal bioactive fragment of nociceptin. |
| M52961 | Ac-RYYRIK-NH2 | Ac-RYYRIK-NH2 is a potent and partial agonist on ORL1 transfected in CHO cells (Kd=1.5 nM) and behaves as a endogenous ligand of ORL1. |
| M52960 | Deltakephalin | Deltakephalin is a potent, selective opiate δ-receptor agonist. |
| M52959 | Biphalin TFA | Biphalin TFA, a BBB-penetrable opioid peptide analog, contains two active enkephalin pharmacophores. |
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