| Cat.No. | Name | Information |
|---|---|---|
| M4808 | TRV130 hydrochloride | TRV130 (Oliceridine) hydrochloride is a novel μ-opioid receptor (MOR) G protein-biased ligand. |
| M1579 | Naloxone | Naloxone is an opioid inverse agonist drug used to counter the effects of opiate overdose. |
| M9615 | DAMGO | DAMGO is an opioid receptor agonist with the ability to affect the locomotive activity in rodents, Kd value is 3.46 nM for native μ-OPR. |
| M28027 | Enadoline | Enadoline (CI-977) is a highly selective, brain-penetrating, and nonpeptide kappa-opioid receptor (KOR) agonist (Ki=1.25 nM). Antinociceptive effects. |
| M27965 | TAN-67 dihydrobromide | TAN-67 (SB-205607) dihydrobromide is a potent and selective nonpeptidic δ-opioid receptor agonist with a Ki value of 0.647 nM. TAN-67 dihydrobromide has neuroprotective effect. TAN-67 dihydrobromide can be used in research of ischemic stroke. |
| M27962 | MT-7716 hydrochloride | MT-7716 hydrochloride (W-212393 hydrochloride) is a selective non-peptide nociceptin receptor (NOP) agonist and promising potential treatment drug for alcohol abuse and relapse prevention. |
| M27855 | ICI 199441 | ICI 199441 is a potent and selective κ-opioid receptor agonist. ICI 199441 can improve heart resistance to ischemia/reperfusion. |
| M21657 | Bevenopran | Bevenopran (CB-5945) is a peripheral μ-opioid receptor antagonist. |
| M21375 | BMS-986187 | BMS-986187 is a δ-opioid receptor selective orthosteric modulator (PAM) with an EC50 of 0.03 μM and a pKB of 6.02 (~1 μM). bms-986187 has no observable PAM activity at the μ receptor (EC50=3 μM). |
| M21363 | TRV-130 | TRV 130 is a novel μ-opioid receptor (MOR) G protein-biased ligand; elicits robust G protein signaling(pEC50=8.1), with potency and efficacy similar to morphine, but with far less β-arrestin recruitment and receptor internalization. |
| M21317 | EST73502 | EST73502 is a selective, orally active, μ-opioid receptor (μ-opioid receptor/MOR) agonist and σ1 receptor (σ1R) antagonist that crosses the blood-brain barrier with Ki values of 64 nM and 118 nM for MOR and σ1R effects, respectively. EST73502 can be used in pain relief studies. |
| M20425 | (-)-Menthol | (-)-Menthol is a levo isomer of menthol and used as a cooling agent that strongly activates TRPM8. |
| M14033 | Ro 64-6198 | Ro 64-6198 is a potent, selective, nonpeptide, high-affinity, high cellular permeability and brain penetration N/OFQ receptor (NOP) agonist with an EC50 value of 25.6 nM. |
| M14032 | Norbinaltorphimine dihydrochloride | Norbinaltorphimine dihydrochloride is a potent and selective κ opioid receptor antagonist. |
| M10564 | CYT-1010 | CYT-1010 is a mu-opioid receptor agonist with EC50s of 13.1 nM and 0.0053 nM on beta-arrestin recruitment and inhibition of cAMP production, respectively. |
| M8832 | U-69593 | U-69593 is a selective κ opioid receptor agonist. |
| M7267 | SB 612111 hydrochloride | SB 612111 hydrochloride is a selective NOP receptor antagonist. |
| M7035 | NNC 63-0532 | NNC 63-0532 is a potent non-peptide NOP agonist; brain penetrant. |
| M7012 | Naloxone benzoylhydrazone | Naloxone benzoylhydrazone is a full κ agonist, partial μ and δ agonist and antagonizes agonist-induced activation of NOP. |
| M3240 | MCOPPB trihydrochloride | MCOPPB trihydrochloride is a trihydrochloride form of MCOPPB that is a new nonpeptide nociceptin/orphanin FQ peptide (NOP)-receptor agonist with a pKi of 10.07 ±0.01 for the human NOP recepto |
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