Free shipping on all orders over $ 500

NNC 63-0532

Cat. No. M7035

All AbMole products are for research use only, cannot be used for human consumption.

NNC 63-0532 Structure

Price and Availability

For this product's availability, delivery time and price, please email [email protected] directly or click the "Inquiry Now" button below.


Quality Control & Documentation
Biological Activity

NNC 63-0532 is a potent non-peptide agonist for the NOP receptor (EC50 = 305 nM, Ki = 7.3 nM); ~ 12-fold selective over other receptors. Centrally active following systemic administration in vivo.

Chemical Information
Molecular Weight 443.54
Formula C27H29N3O3
CAS Number 250685-44-0
Solubility (25°C) DMSO 22.18 mg/mL
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Willems, et al. Cell Stem Cell. Small molecule-mediated TGF-beta type II receptor degradation promotes cardiomyogenesis in embryonic stem cells.

Related Opioid Receptor Products
SNC162 

SNC162 is a delta-opioid receptor agonist with an IC50 of 0.94 nM.

ML 190 

ML 190 is a selective κ opioid receptor (KOR) antagonist with an IC50 of 120 nM and an EC50 of 129 nM, respectively.

CCG258747 

CCG258747 is a selective GRK2 inhibitor (IC50=18 nM) with high selectivity over GRK1, GRK5, PKA, and ROCK1 (518, 83, >5500, and >550–fold, respectively).CCG258747 also blocks the internalization of the µ-opioid receptor.

Sunobinop

Sunobinop (S 117957) is a modulator of the opioid receptor-like orphan receptor (ORL1).

SCH 486757 

SCH 486757 is an orally effective pain peptide receptor (NOP) agonist.

  Catalog
Abmole Inhibitor Catalog




Keywords: NNC 63-0532 supplier, Opioid Receptor, inhibitors, activators

All AbMole products are for research use only, cannot be used for human consumption or veterinary use. We do not provide products or services to individuals. Please comply with the intended use and do not use AbMole products for any other purpose.



Products are for research use only. Not for human use. We do not sell to patients.
© Copyright 2010-2024 AbMole BioScience. All Rights Reserved.