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CTOP TFA is a peptide that acts as a potent and selective μ opioid receptor antagonist, with Ki values of 0.96 and >10,000 nM for μ and δ receptors, respectively. CTOP TFA increases K+ currents in rat locus ceruleus neurons in vitro via a μ receptor independent mechanism.
| Molecular Weight | 1176.28 |
| Formula | C52H68F3N11O13S2 |
| CAS Number | 103429-31-8 (free base) |
| Solubility (25°C) | Water 45 mg/mL |
| Storage | -20°C, protect from light, sealed |
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