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Dynorphin A (1-8) is the most likely natural ligand of the kappa receptor. Dynorphin A (1-8) inhibited 3H-Bremazocine binding to the purified kappa receptor with IC50 of 303 nM. Dynorphin A (1-8) is an opioid octapeptide that exhibits agonist activity at μ and δ receptors.
| Molecular Weight | 981.15 |
| Formula | C46H72N14O10 |
| CAS Number | 75790-53-3 |
| Storage |
Powder -20°C 3 years ; 4°C 2 years In solvent -80°C 6 months ; -20°C 1 month |
| Related Opioid Receptor Products |
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ML 190 is a selective κ opioid receptor (KOR) antagonist with an IC50 of 120 nM and an EC50 of 129 nM, respectively. |
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| Sunobinop
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| SCH 486757
SCH 486757 is an orally effective pain peptide receptor (NOP) agonist. |
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