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SR17018

Cat. No. M10584

All AbMole products are for research use only, cannot be used for human consumption.

SR17018 Structure
Synonym:

SR-17018

Size Price Availability Quantity
5mg USD 80  USD80 In stock
10mg USD 130  USD130 In stock
25mg USD 260  USD260 In stock
50mg USD 420  USD420 In stock
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Quality Control & Documentation
Biological Activity

SR17018 is an mu-opioid-receptor (MOR) agonist with an EC50 of 97 nM. SR17018 promotes signaling through G proteins or βarrestin2.

Chemical Information
Molecular Weight 410.72
Formula C19H18Cl3N3O
CAS Number 2134602-45-0
Solubility (25°C) DMSO 10 mg/mL
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Cullen L Schmid, et al. Cell. Bias Factor and Therapeutic Window Correlate to Predict Safer Opioid Analgesics

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Keywords: SR17018, SR-17018 supplier, Opioid Receptor, inhibitors, activators

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