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 About 30 results found for searched term "Dopamine Receptor" (0.044 seconds)

Cat.No.  Name Target
M2349 (R)-Nepicastat hydrochloride HCV Protease
RS-25560-198 HCl
(R)-Nepicastat hydrochloride, the R-enantiomer of Nepicastat hydrochloride, is a potent and selective inhibitor with IC50 of 25.1 nM and 18.3 nM for bovine and human dopamine-β-hydroxylase, with negligible affinity for twelve other enzymes and thirteen neurotransmitter receptors.
M2372 Alizapride hydrochloride Dopamine Receptor
Alizapride hydrochloride is a dopamine receptor antagonist used for the theropy of nausea and vomiting.
M2445 Benztropine mesylate Dopamine Receptor
Benzatropine mesylate; Benzotropine mesylate; Benztropine methanesulfonate
Benztropine is a dopamine transporter (DAT) inhibitor with IC50 of 118 nM. Benztropine mesylate is a human D2 dopamine receptor allosteric antagonist. Benztropine mesylate also has anti-CSCs (cancer stem cells) effects. Benztropine mesylate is also an anti-histamine agent and a dopamine re-uptake inhibitor.
M2494 Cariprazine hydrochloride Dopamine Receptor
RGH-188 HCl
Cariprazine hydrochloride is a dopamine D3-receptor-preferring partial agonist that exhibits high selectivity and affinity to dopamine D3 and D2(L/S) receptors with pKi 10.07 and 9.16/9.31, respectively.
M2655 Droperidol Dopamine Receptor
Dehydrobenzperidol
Droperidol is a potent antagonist of dopamine subtype 2 receptors in the limbic system.
M2886 Nomifensine Maleate Dopamine Receptor
(±)-Nomifensine maleat
Nomifensine is a dopamine reuptake inhibitor that increases the amount of synaptic dopamine available to receptors by blocking dopamine's re-uptake transporter.
M2925 Pergolide mesylate Dopamine Receptor
LY127809
Pergolide mesylate is a potent and orally active dopamine D1 and D2 receptors agonist. Pergolide mesylate can be used for the research of Parkinson's disease and hyperprolactinaemia.
M2936 Phenothiazine Dopamine Receptor
Phenothiazine is a dopamine-2 (D2) receptor antagonist therefore decreases the effect of dopamine in the brain.
M2987 Ropinirole hydrochloride Dopamine Receptor
SKF 101468 hydrochloride
Ropinirole a selective dopamine D2 receptors inhibitor with IC50 of 29 nM.
M3065 Thioridazine hydrochloride Dopamine Receptor
Thioridazine is a trifluoro-methyl phenothiazine derivative, which blocks postsynaptic mesolimbic dopaminergic D1 and D2 receptors in the brain.
M3087 Trifluoperazine dihydrochloride Dopamine Receptor
TFP; SKF5019
Trifluoperazine is a dopamine D2 receptor inhibitor with IC50 of 1.1 nM.
M3088 Triflupromazine hydrochloride Dopamine Receptor
Triflupromazine hydrochloride is a member of a family of phenothiazine compounds that are dopamine D1/D2 receptor antagonists.
M3165 Prochlorperazine dimaleate Dopamine Receptor
Prochlorperazine dimaleate is a D2 dopamine receptor antagonist.
M3242 Sumanirole Maleate Dopamine Receptor
U 95666E
Sumanirole maleate is a highly selective dopamine D2 receptor agonist with binding affinity of 9 nM and EC50 of about 46 nM, exhibits >200-fold selectivity over the other dopamine receptor subtypes.
M3287 PD128907 hydrochloride Dopamine Receptor
PD 128907 hydrochloride is a potent and selective dopamine D3 receptor agonist, with EC50 of 0.64 nM, exhibits 53-fold selectivity over dopamine D2 receptor.
M3320 Quetiapine Fumarate 5-HT Receptor
Quetiapine hemifumarate
Quetiapine hemifumarate is a 5-HT receptors agonist with a pEC50 of 4.77 for human 5-HT1A receptor. Quetiapine hemifumarate is a dopamine receptor antagonist with a pIC50 of 6.33 for human D2 receptor.
M3414 Olanzapine 5-HT Receptor
LY170053
Olanzapine is a high affinity for 5-HT2 serotonin and D2 dopamine receptor antagonist.
M3479 Aripiprazole 5-HT Receptor
OPC-14597
Aripiprazole is a human 5-HT1A receptor partial agonist with a Ki of 4.2 nM. Aripiprazole (OPC-14597) is a potent and high-affinity dopamine D2 receptor partial agonist.
M3481 WAY-100635 Maleate 5-HT Receptor
WAY-100635 maleate is a potent, selective 5-HT1A receptor antagonist with an IC50 value of 0.91 nM, a Ki value of 0.39 nM, and a pIC50 of 8.87, which is more than 100-fold more selective than for use at the other 5-HT receptor subtypes and major neurotransmitter receptors. In addition, WAY-100635 maleate is a potent dopamine D4 receptor agonist.
M3592 Chlorprothixene Dopamine Receptor
Chlorprothixene has strong binding affinities to dopamine and histamine receptors, such as D1, D2, D3, D5, H1, 5-HT2, 5-HT6 and 5-HT7, with Ki of 18 nM, 2.96 nM, 4.56 nM, 9 nM, 3.75 nM, 9.4 nM, 3 nM and 5.6 nM, respectively.
M3670 Metoclopramide hydrochloride 5-HT Receptor
Metoclopramide hydrochloride is a selective dopamine D2 receptor antagonist, used for the treatment of nausea and vomiting.
M3674 Metoclopramide Dopamine Receptor
Metoclopramide is a potent antagonist of 5-HT3 and dopamine D2 receptor, with IC50s of 308 nM and 483 nM, respectively.
M3675 Rotigotine Dopamine Receptor
N-0923; (-)-N 0437
Rotigotine is a potent dopamine receptor agonist with Ki values of 0.71 nM, 4-15 nM, and 83 nM for the dopamine D3 receptor and D2, D5, D4 receptors and dopamine D1 receptor. Rotigotine a partial agonist of the 5-HT1A receptor, and an antagonist of the α2B-adrenergic receptor.
M3785 Flupenthixol dihydrochloride Dopamine Receptor
Flupenthixol 2HCl
Flupenthixol dihydrochloride is a dopamine receptor antagonist which acts as a Neuroleptic agent as well as an antipsychotic.
M3818 Rotigotine Hydrochloride Dopamine Receptor
Rotigotine HCl;N-0923 Hydrochloride
Rotigotine Hydrochloride (N-0923 Hydrochloride) is a full agonist of dopamine receptor, a partial agonist of the 5-HT1A receptor, and an antagonist of the α2B-adrenergic receptor, with Ki of 0.71 nM, 4-15 nM, and 83 nM for the dopamine D3 receptor and D2, D5, D4 receptors, and dopamine D1 receptor.
M1565 Quetiapine sulfoxide 5-HT Receptor
Quetiapine sulfoxide; Quetiapine S-oxide
Quetiapine sulfoxide is a 5-HT receptor agonist with a pEC50 value of 4.77 for human 5-HT1A. Quetiapine hemifumarate is a dopamine receptor antagonist with a pIC50 value of 6.33 for human D2.
M1564 Quetiapine Sulfone 5-HT Receptor
Quetiapine Sulfone is a 5-HT receptor agonist with a pEC50 value of 4.77 for human 5-HT1A. Quetiapine hemifumarate is a dopamine receptor antagonist with a pIC50 value of 6.33 for human D2.
M1454 Buspirone 5-HT Receptor
Buspirone is an orally active 5-HT1A receptor agonist, and a dopamine D2 autoreceptorsant antagonist.
M4458 Tetrahydroberberine Dopamine Receptor
Canadine; THB
Tetrahydroberberine is an isoquinoline alkaloid isolated from corydalis tuber; has micromolar affinity for dopamine D(2) (pK(i) = 6.08) and 5-HT(1A) (pK(i) = 5.38) receptors but moderate to no affinity for other relevant serotonin receptors (5-HT(1B), 5-HT(1D), 5-HT(3), and 5-HT(4); pK(i) < 5.00).
M4887 Pardoprunox Hydrochloride 5-HT Receptor
SLV-308
Pardoprunox hydrochloride (DU-126891, SME-308) is an effective agonist of partial dopamine action, corresponding to pEC50 value 8.0. It is also a partial agonist inducing [35S]GTPγS binding, corresponding to pEC50 9.2 and serotonin 5-HT1A receptor 6.3.



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