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Quetiapine Fumarate

Cat. No. M3320

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Quetiapine Fumarate Structure
Synonym:

Quetiapine hemifumarate

Size Price Availability Quantity
Free Sample (0.5-1 mg)  USD 0 In stock
100mg USD 30  USD30 In stock
500mg USD 50  USD50 In stock
1g USD 60  USD60 In stock
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Quality Control & Documentation
Biological Activity

Quetiapine hemifumarate is a 5-HT receptors agonist with a pEC50 of 4.77 for human 5-HT1A receptor. Quetiapine hemifumarate is a dopamine receptor antagonist with a pIC50 of 6.33 for human D2 receptor.

Chemical Information
Molecular Weight 883.09
Formula C46H54N6O8S2
CAS Number 111974-72-2
Solubility (25°C) DMSO 25 mg/mL
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Michael Poyurovsky, et al. Low-Dose Quetiapine Fumarate (50 mg) for Obsessive-Compulsive Disorder Patients With Comorbid Bipolar Depression

[2] Shweta Agarwal, et al. Quetiapine Fumarate Loaded Nanostructured Lipid Carrier for Enhancing Oral Bioavailability: Design, Development and Pharmacokinetic Assessment

[3] Karen Astrid Boldingh Debernard, et al. Quetiapine is not a sleeping pill

[4] N El-Saifi, et al. Quetiapine safety in older adults: a systematic literature review

[5] Sirijit Suttajit, et al. Quetiapine for acute bipolar depression: a systematic review and meta-analysis

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Keywords: Quetiapine Fumarate, Quetiapine hemifumarate supplier, 5-HT Receptor, inhibitors, activators

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