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5-HT Receptor 5-hydroxytryptamine receptor

Inhibitors

Cat.No.  Name Information
M2048 Sumatriptan succinate Sumatriptan succinate is a 5-HT1 serotonin receptor agonist.
M3417 Clozapine Clozapine is a potent 5-HT1C receptor antagonist with an IC50 of 110 nM for 5-HT-stimulated phosphoinositide hydrolysis.
M3985 Triptolide Triptolide is a structurally unique diterpene triepoxide isolated from a traditional Chinese medicinal plant with anti-inflammatory, immunosuppressive, contraceptive and antitumor activities.
M2821 Lorcaserin hydrochloride Lorcaserin hydrochloride is a selective full agonist of human 5-HT2C receptor with Ki of 15 nM.
M10779 Alniditan dihydrochloride Anidetam dihydrochloride Alniditan (Alnitidan) dihydrochloride is an effective one 5-HT1B and 5-HT1D RECEPTOR AGONISTS, IN HEK 293 CELLS, IN HUMANS 5-HT1B and people 5-HT1D receptors IC50 1.7 nM and 1.3 nM, respectively. Alniditan dihydrochloride has the effect of preventing migraines.
M10608 NLX-101 (F-15599) NLX-101 (F-15599) is a highly selective G-protein biased 5-HT1A receptor agonist, with Ki of 3.4 nM. NLX-101 (F-15599) mediates antidepressant-like activity in rats via prefrontal cortex 5-HT 1A receptors. NLX-101 (F-15599) has over 1000-fold higher affinity for this target over other receptors.
M10345 Eucalyptol Eucalyptol is an inhibitor of 5-HT3 receptor, potassium channel, with anti-inflammatory and antioxidant activities.
M10160 Lasmiditan Lasmiditan (COL-144; LY573144) is a novel, centrally acting, highly selective 5-HT(1F) receptor agonist, showed a K(i) value of 2.21 nM at the 5-HT(1F) receptor in vitro binding studies.
M10054 Paroxetine Paroxetine is a inhibitor of serotonin uptake.
M9763 AVN-492 AVN-492 is a potent and selective 5-HT6R antagonist, binds to 5-HT6R (Ki = 91 pM).
M9584 SAM-315 SAM-31 (WAY-255315) is selective 5-Hydroxytryptamine-6 antagonists.
M9565 RU 24969 hemisuccinate RU 24969 hemisuccinate is a selective agonist at the 5-HT1A and 5-HT1B receptors.
M9308 LY344864 LY344864 is a selective 5-HT1F receptor agonist with an affinity of 6 nM (Ki).
M9252 YL-0919 YL-0919 is a novel 5-HT1A receptor agonist and selective serotonin reuptake inhibitor.
M9181 8-OH-DPAT 8-OH-DPAT (8-Hydroxy-DPAT) is a potent and selective 5-HT agonist, with a pIC50 of 8.19 for 5-HT1A.
M9025 Idalopirdine hydrochloride Idalopirdine hydrochloride is a potent and selective 5-HT6 receptor antagonist with a Ki value of 0.83 nM.
M9011 PRX-08066 PRX-08066 is a a novel 5-hydroxytryptamine receptor 2B antagonist with IC50 of 3.4 nM.
M8955 MIN-101 MIN-101 (Roluperidone) is a novel compound with affinities for 5-HT2A and sigma-2 receptors with Ki values of 7.53 nM and 8.19 nM, respectively.
M8942 GSK163090 GSK163090 is a potent, selective, and orally active 5-HT1A/B/D receptor antagonist.
M8932 Eptapirone Eptapirone (F11440) is a potent 5HT(1A) receptor agonist with marked anxiolytic and antidepressant potential.
M8900 TG6-10-1 TG6-10-1 is a potent and selective antagonist for the prostaglandin E2 receptor subtype EP2.
M8856 WAY-100135 dihydrochloride WAY-100135 dihydrochloride is a potent, selective 5-HT1A receptor antagonist (IC50 = 15 nM).
M8033 Paroxetine hydrochloride hemihydrate Paroxetine hydrochloride hemihydrate is one of the most potent and selective of the selective serotonin reuptake inhibitors (SSRI); antidepressant.
M7684 Clozapine N-oxide Clozapine N-oxide (CNO) is a 5-HT2 serotonin receptor antagonist; major metabolite of clopazine that can be monitored by HPLC.



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