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Inhibitors
| Cat.No. | Name | Information |
|---|---|---|
| M2048 | Sumatriptan succinate | Sumatriptan succinate is a 5-HT1 serotonin receptor agonist. |
| M3417 | Clozapine | Clozapine is a potent 5-HT1C receptor antagonist with an IC50 of 110 nM for 5-HT-stimulated phosphoinositide hydrolysis. |
| M3985 | Triptolide | Triptolide is a structurally unique diterpene triepoxide isolated from a traditional Chinese medicinal plant with anti-inflammatory, immunosuppressive, contraceptive and antitumor activities. |
| M2821 | Lorcaserin hydrochloride | Lorcaserin hydrochloride is a selective full agonist of human 5-HT2C receptor with Ki of 15 nM. |
| M10779 | Alniditan dihydrochloride | Anidetam dihydrochloride Alniditan (Alnitidan) dihydrochloride is an effective one 5-HT1B and 5-HT1D RECEPTOR AGONISTS, IN HEK 293 CELLS, IN HUMANS 5-HT1B and people 5-HT1D receptors IC50 1.7 nM and 1.3 nM, respectively. Alniditan dihydrochloride has the effect of preventing migraines. |
| M10608 | NLX-101 (F-15599) | NLX-101 (F-15599) is a highly selective G-protein biased 5-HT1A receptor agonist, with Ki of 3.4 nM. NLX-101 (F-15599) mediates antidepressant-like activity in rats via prefrontal cortex 5-HT 1A receptors. NLX-101 (F-15599) has over 1000-fold higher affinity for this target over other receptors. |
| M10345 | Eucalyptol | Eucalyptol is an inhibitor of 5-HT3 receptor, potassium channel, with anti-inflammatory and antioxidant activities. |
| M10160 | Lasmiditan | Lasmiditan (COL-144; LY573144) is a novel, centrally acting, highly selective 5-HT(1F) receptor agonist, showed a K(i) value of 2.21 nM at the 5-HT(1F) receptor in vitro binding studies. |
| M10054 | Paroxetine | Paroxetine is a inhibitor of serotonin uptake. |
| M9763 | AVN-492 | AVN-492 is a potent and selective 5-HT6R antagonist, binds to 5-HT6R (Ki = 91 pM). |
| M9584 | SAM-315 | SAM-31 (WAY-255315) is selective 5-Hydroxytryptamine-6 antagonists. |
| M9565 | RU 24969 hemisuccinate | RU 24969 hemisuccinate is a selective agonist at the 5-HT1A and 5-HT1B receptors. |
| M9308 | LY344864 | LY344864 is a selective 5-HT1F receptor agonist with an affinity of 6 nM (Ki). |
| M9252 | YL-0919 | YL-0919 is a novel 5-HT1A receptor agonist and selective serotonin reuptake inhibitor. |
| M9181 | 8-OH-DPAT | 8-OH-DPAT (8-Hydroxy-DPAT) is a potent and selective 5-HT agonist, with a pIC50 of 8.19 for 5-HT1A. |
| M9025 | Idalopirdine hydrochloride | Idalopirdine hydrochloride is a potent and selective 5-HT6 receptor antagonist with a Ki value of 0.83 nM. |
| M9011 | PRX-08066 | PRX-08066 is a a novel 5-hydroxytryptamine receptor 2B antagonist with IC50 of 3.4 nM. |
| M8955 | MIN-101 | MIN-101 (Roluperidone) is a novel compound with affinities for 5-HT2A and sigma-2 receptors with Ki values of 7.53 nM and 8.19 nM, respectively. |
| M8942 | GSK163090 | GSK163090 is a potent, selective, and orally active 5-HT1A/B/D receptor antagonist. |
| M8932 | Eptapirone | Eptapirone (F11440) is a potent 5HT(1A) receptor agonist with marked anxiolytic and antidepressant potential. |
| M8900 | TG6-10-1 | TG6-10-1 is a potent and selective antagonist for the prostaglandin E2 receptor subtype EP2. |
| M8856 | WAY-100135 dihydrochloride | WAY-100135 dihydrochloride is a potent, selective 5-HT1A receptor antagonist (IC50 = 15 nM). |
| M8033 | Paroxetine hydrochloride hemihydrate | Paroxetine hydrochloride hemihydrate is one of the most potent and selective of the selective serotonin reuptake inhibitors (SSRI); antidepressant. |
| M7684 | Clozapine N-oxide | Clozapine N-oxide (CNO) is a 5-HT2 serotonin receptor antagonist; major metabolite of clopazine that can be monitored by HPLC. |
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