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Vabicaserin hydrochloride

Cat. No. M55224

All AbMole products are for research use only, cannot be used for human consumption.

Vabicaserin hydrochloride Structure
Synonym:

SCA 136

Size Price Availability Quantity
1mg USD 155  USD155 In stock
5mg USD 380  USD380 In stock
10mg USD 540  USD540 In stock
25mg USD 850  USD850 In stock
50mg USD 1200  USD1200 In stock
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Quality Control & Documentation
Biological Activity

Vabicaserin hydrochloride is a 5-hydroxytryptamine 2C (5-HT2C) receptor-selective agonist with an EC50 of 8 nM. Vabicaserin exhibits lower affinity at the 5-HT2C antagonist binding site (22 nM) labeled with [3H]mesulergine. Additional binding studies indicate that Vabicaserin possesses affinity for the 5-HT2B and 5-HT1A receptors with Ki values of 14 and 112 nM, respectively.

Chemical Information
Molecular Weight 264.79
Formula C15H21ClN2
CAS Number 887258-94-8
Solubility (25°C) DMSO 60 mg/mL
Water 4 mg/mL
Storage 4°C, dry, sealed
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Keywords: Vabicaserin hydrochloride, SCA 136 supplier, 5-HT Receptor, inhibitors, activators

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