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5-HT2B antagonist-1

Cat. No. M58155

All AbMole products are for research use only, cannot be used for human consumption.

5-HT2B antagonist-1 Structure
Size Price Availability Quantity
5mg USD 50  USD50 In stock
10mg USD 80  USD80 In stock
25mg USD 130  USD130 In stock
50mg USD 240  USD240 In stock
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Quality Control & Documentation
Biological Activity

5-HT2B antagonist-1 is an orally active 5-HT2B receptor antagonist with an IC50 value of 33.4 nM.

5-HT2B antagonist-1 (oral gavage, 30 mg/kg) can reduce visceral hypersensitivity significantly in irritable bowel syndrome (IBS) rats.

5-HT2B antagonist-1 can be used in studies of diseases characterized by 5-HT2B receptor signaling, such as hepatocellular carcinoma, cardiovascular disease or gastrointestinal disease.

Chemical Information
Molecular Weight 296.17
Formula C11H14BrN5
CAS Number 393129-91-4
Solubility (25°C) DMSO 30 mg/mL
Water 7 mg/mL
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
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Keywords: 5-HT2B antagonist-1 supplier, 5-HT Receptor, inhibitors, activators

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