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Lorcaserin hydrochloride is a selective full agonist of human 5-HT2C receptor with Ki of 15 nM.
J Clin Invest. 2021 Dec 15;131(24):e151976.
Melanocortin 4 receptor stimulation prevents anti-depressant-associated weight gain in mice caused by long-term fluoxetine exposure
Lorcaserin hydrochloride purchased from AbMole
| Molecular Weight | 232.15 |
| Formula | C11H14ClN.HCl |
| CAS Number | 846589-98-8 |
| Solubility (25°C) | DMSO 26 mg/mL |
| Storage |
Powder -20°C 3 years ; 4°C 2 years In solvent -80°C 6 months ; -20°C 1 month |
[1] Andrea Cignarella, et al. Pharmacotherapy of obesity: An update
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