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Cariprazine hydrochloride

Cat. No. M2494

All AbMole products are for research use only, cannot be used for human consumption.

Cariprazine hydrochloride Structure
Synonym:

RGH-188 HCl

Size Price Availability Quantity
5mg USD 30  USD30 In stock
10mg USD 50  USD50 In stock
25mg USD 75  USD75 In stock
50mg USD 120  USD120 In stock
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Quality Control & Documentation
Biological Activity

Cariprazine hydrochloride is a dopamine D3-receptor-preferring partial agonist that exhibits high selectivity and affinity to dopamine D3 and D2(L/S) receptors with pKi 10.07 and 9.16/9.31, respectively.

Chemical Information
Molecular Weight 463.87
Formula C21H32Cl2N4O.HCl
CAS Number 1083076-69-0
Solubility (25°C) DMSO 6 mg/mL
Water 2 mg/mL
Storage 4°C, dry, sealed
References

[1] No authors listed. Aust Prescr. Cariprazine hydrochloride for schizophrenia

[2] Amber Edinoff, et al. Cariprazine to Treat Schizophrenia and Bipolar Disorder in Adults

[3] Renee-Marie Ragguett, et al. Cariprazine for the treatment of bipolar depression: a review

[4] Lakshmi N Yatham, et al. Canadian Network for Mood and Anxiety Treatments (CANMAT) and International Society for Bipolar Disorders (ISBD) 2018 guidelines for the management of patients with bipolar disorder

[5] Karly P Garnock-Jones. Cariprazine: A Review in Schizophrenia

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Keywords: Cariprazine hydrochloride, RGH-188 HCl supplier, Dopamine Receptor, inhibitors, activators

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