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Inhibitors
| Cat.No. | Name | Information |
|---|---|---|
| M5686 | Haloperidol | Haloperidol is a potent dopamine D2 receptor antagonist. |
| M11167 | A-381393 | A-381393 IS AN EFFECTIVE, SELECTIVE, AND BLOOD-BRAIN BARRIER-PERMEABLE dopamine D4 receptor Antagonist, dopamine D for humans4.4，D4.2 AND D4.7 receptors Ki The values are 1.5, 1.9, and 1.6 nM, respectively, with selectivity being D1，D2，D3，D5 MORE THAN 2700 TIMES THE DOPAMINE RECEPTOR. A-381393 VS. 5-HT2A MODERATE SELECTIVITY, Ki The value is 370 nM. |
| M10724 | Pridopidine | Pridopidine is a dopamine (DA) stabilizer that acts as a low-affinity dopamine D2 receptor (D2R) antagonist. Pridopidine high affinity acts on sigma 1 receptor (S1R),Ki Values of 70 to 80 nM are approximately 100 times higher than their affinity for D2R. |
| M10494 | ML417 | ML417 is a highly selective and brain penetrant D3 dopamine receptor (D3R) agonist, with EC50 of 38 nM. |
| M9601 | Cariprazine | Cariprazine is a D2 and D3 receptor partial agonist, with high selectivity towards the D3 receptor. |
| M9482 | PD-168077 maleate | PD-168077 maleate is a potent D4 dopamine receptor agonist (Ki = 8.7 nM), with > 400-fold and > 300-fold selectivity over D2 / D3 subtypes, respectively. |
| M9099 | SCH23390 | SCH23390 is a potent dopamine receptor antagonist (Ki values are 0.2 nM and 0.3 nM at D1 and D5 receptor sub-types, respectively). |
| M9049 | MPTP HCl | MPTP hcl is a compound to the neurotoxin MPP+ which causes permanent symptoms of Parkinson's disease. |
| M9022 | SKF38393 HCl | SKF38393 HCl is a selective D1 dopamine receptor agonist with IC50 of 110 nM. |
| M7832 | 6-Hydroxydopamine hydrochloride | 6-Hydroxydopamine hydrochloride is an antagonist of the neurotransmitter dopamine. |
| M7279 | SCH 23390 hydrochloride | SCH 23390 hydrochloride is a standard selective D 1-like antagonist; also 5-HT 2C and 5-HT 1C agonist and K ir3 channel blocker. |
| M5984 | Sulpiride | Sulpiride is a dopamine D2-receptor antagonist. It has been used therapeutically as an antidepressant, antipsychotic, and as a digestive aid. |
| M5914 | rac-Rotigotine (Hydrochloride) | rac-Rotigotine Hcl is a high potency and selectivity agonist for D-2 receptor with Ki of 0.69 nM. |
| M5903 | Promazine HCl | Promazine (hydrochloride) is a D2 dopamine receptor antagonist, belongs to the phenothiazine class of antipsychotics, used to treat schizophrenia. |
| M5900 | Prochlorperazine dimaleate salt | Prochlorperazine dimaleate is a dopamine (D2) receptor antagonist. |
| M5891 | Pramipexole dihydrochloride | Pramipexole 2Hcl is a partial/full D2S, D2L, D3, D4 receptor agonist with a Ki of 3.9, 2.2, 0.5 and 5.1 nM for D2S, D2L, D3, D4 receptor, respectively. |
| M5872 | Perphenazine | Perphenazine is a phenothiazine derivative and a dopamine antagonist with antiemetic and antipsychotic properties. |
| M5854 | SB 277011 Hydrochloride | Ligands acting as DRD3 antagonists (SB 277011-A) has shown some promise for reducing the influence of drug-associated cues on motivational behaviour. |
| M5848 | Paliperidone | Paliperidone, the main active metabolite of Risperidone, is a potent serotonin-2A and dopamine-2 receptor antagonist, used in the treatment of schizophrenia. |
| M5796 | Molindone HCl | Molindone is an antipsychotic compound used to study schizophrenia that reduces psychosis by blocking the action of dopamine in the brain. |
| M5739 | Levosulpiride | Levosulpiride is a selective antagonist for D2 dopamine receptors used as an antipsychotic and prokinetic agent. |
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