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Dopamine Receptor Dopamine Receptor

Inhibitors

Cat.No.  Name Information
M5686 Haloperidol Haloperidol is a potent dopamine D2 receptor antagonist.
M5410 Amisulpride Amisulpride is an atypical antipsychotic used to treat psychosis in schizophrenia and episodes of mania in bipolar disorder.
M5350 (+,-)-Octopamine Octopamine (OA), a biogenic monoamine structurally related to noradrenaline, acts as a neurohormone, a neuromodulator and a neurotransmitter in invertebrates.
M5198 Fluphenazine dihydrochloride Fluphenazine dihydrochloride is a phenothiazine-class D1DR and D2DR inhibitor.
M4942 Metoclopramide hydrochloride hydrate Metoclopramide hydrochloride hydrate is a dopamine D2 antagonist that is used as an antiemetic.
M3818 Rotigotine Hydrochloride Rotigotine Hydrochloride (N-0923 Hydrochloride) is a pure agonist of the dopamine receptor, a partial agonist of the 5-HT1A receptor, and an antagonist of the α2B-adrenergic receptor.Ki 值分别为 0.71 nM (dopamine D3 receptor),4-15 nM (D2,D5,D4 receptors),83 nM (dopamine D1 receptor)。
M3785 Flupenthixol dihydrochloride Flupenthixol dihydrochloride is a dopamine receptor antagonist which acts as a Neuroleptic agent as well as an antipsychotic.
M3675 Rotigotine Rotigotine (N-0437; N-0923) is a dopamine receptor agonist, a partial agonist of the 5-HT1A receptor, and an antagonist of the α2B-adrenergic receptor.Ki 值分别为 0.71 nM (dopamine D3 receptor),4-15 nM (D2,D5,D4 receptors),83 nM (dopamine D1 receptor)。
M3674 Metoclopramide Metoclopramide is a dopamine D2 antagonist that is used as an antiemetic.
M3586 Pramipexole dihydrochloride Monohydrate Pramipexole dihydrochloride Monohydrate is a partial/full D2S, D2L, D3, D4, receptor agonist with a Ki of 3.9, 2.2, 0.5, 5.1 nM.
M3338 Domperidone Domperidone is a dopamine blocker and an antidopaminergic reagent.
M3287 PD128907 hydrochloride PD 128907 hydrochloride is a potent and selective dopamine D3 receptor agonist, with EC50 of 0.64 nM, exhibits 53-fold selectivity over dopamine D2 receptor.
M3250 Vanoxerine dihydrochloride Vanoxerine dihydrochloride (GBR-12909 dihydrochloride) is a potent and selective dopamine receptor inhibitor.
M3246 Amfebutamone hydrochloride Amfebutamone hydrochloride is a selective norepinephrine-dopamine reuptake inhibitor with IC50 of 6.5 and 3.4μM for the reuptake of dopamine and norepinephrine, respectively
M3242 Sumanirole Maleate Sumanirole maleate is a highly selective dopamine D2 receptor agonist with binding affinity of 9 nM and EC50 of about 46 nM, exhibits >200-fold selectivity over the other dopamine receptor subtypes.
M3165 Prochlorperazine dimaleate Prochlorperazine dimaleate is a D2 dopamine receptor antagonist.
M3088 Triflupromazine hydrochloride Triflupromazine hydrochloride is a member of a family of phenothiazine compounds that are dopamine D1/D2 receptor antagonists.
M3087 Trifluoperazine dihydrochloride Trifluoperazine is a dopamine D2 receptor inhibitor with IC50 of 1.1 nM.
M2987 Ropinirole hydrochloride Ropinirole a selective dopamine D2 receptors inhibitor with IC50 of 29 nM.
M2945 Pimozide Pimozide is an antagonist of 6-hydroxyapatide against 6-hydroxyapatide, with Ki values of 1.4 nM, 2.5 nM and 588 nM for 6-hydroxyapatide, D3 and D1 receptors, respectively. Pimozide also has a high affinity for α1-adrenoceptor. Ki value is 39 nM. Pimozide is also an inhibitor of STAT3 and STAT5, and piperimidate triggers ADCD in glioblastoma cell lines (LN-229, MZ-54, GOS-3 and U343) by inducing dephosphorylation and inactivation of mTORC1.
M2936 Phenothiazine Phenothiazine is a dopamine-2 (D2) receptor antagonist therefore decreases the effect of dopamine in the brain.



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