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Tavapadon

Cat. No. M28766

All AbMole products are for research use only, cannot be used for human consumption.

Tavapadon Structure
Synonym:

PF-06649751; CVL-751

Size Price Availability Quantity
1mg USD 90  USD90 In stock
5mg USD 200  USD200 In stock
10mg USD 300  USD300 In stock
25mg USD 540  USD540 In stock
50mg USD 710  USD710 In stock
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Quality Control & Documentation
Biological Activity

Tavapadon (PF-06649751) is a potentially best-in-class, orally active, highly selective dopamine D1/D5 receptor partial agonist for studies related to Parkinson's disease (PD).

Chemical Information
Molecular Weight 391.34
Formula C19H16F3N3O3
CAS Number 1643489-24-0
Storage Please store the product under the recommended conditions in the Certificate of Analysis.
References

[1] Mechelle M Lewis, et al. Biomolecules. Dopamine D1 Agonists: First Potential Treatment for Late-Stage Parkinson's Disease

[2] Erwan Bezard, et al. CNS Neurol Disord Drug Targets. Rationale and Development of Tavapadon, a D1/D5-Selective Partial Dopamine Agonist for the Treatment of Parkinson's Disease

[3] Xiao Teng, et al. Nat Commun. Ligand recognition and biased agonism of the D1 dopamine receptor

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Keywords: Tavapadon, PF-06649751; CVL-751 supplier, Dopamine Receptor, inhibitors, activators

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