Free shipping on all orders over $ 500

TRP Channel Transient Receptor Potential Channel

Cat.No.  Name Information
M6494 BCTC BCTC is a tRPV1 antagonist. BCTC is also a potent and specific inhibitor of transient receptor potential cation channel subfamily M member 8 (TRPM8) in prostate cancer (PCa) DU145 cells.
M3422 Capsaicin Capsaicin is an active component of chili peppers, which are plants belonging to the genus Capsicum.
M7698 Capsazepine Capsazepine is a specific vanilloid receptor antagonist; synthetic analog of capsaicin.
M10315 MK6-83 MK6-83 is an agonist of the transient receptor potential channel ML3 (TRPML3).
M9962 Nonivamide Nonivamide (also called pelargonic acid vanillylamide or PAVA) can activate the TRPV1 receptor, thus, stimulate the firing rate of dopaminergic neurons in the ventral tegmental area of the brain and to increase the expression of the serotonin receptor gene HTR2A.
M2960 Probenecid Probenecid is a classical competitive inhibitor of organic anion transport, which is also a TRPV2 agonist and an inhibitor of TAS2R16.
M7816 GSK1016790A GSK1016790A is a novel and potent TRPV4 channel agonist.
M7199 RN 1734 RN 1734 is a selective TRPV4 antagonist.
M6983 ML SA1 ML SA1 is a activator of TRPML channels.
M6741 Gadolinium chloride Gadolinium chloride is a stretch-activated calcium channel blocker; calcium-sensing receptor agonist.
M6705 EIPA EIPA (L593754) is an orally active TRPP3 channel inhibitor with an IC50 of 10.5 μM. EIPA also enhances autophagy by inhibiting Na+/H+-exchanger 3 (NHE3).
M6605 CIM 0216 CIM 0216 is a selective TRPM3 agonist.
M6470 ASP7663 ASP7663 is an orally active and selective TRPA1 agonist.
M6441 AMTB hydrochloride AMTB hydrochloride is a tRPM8 blocker.
M6437 AMG 9810 AMG 9810 is a potent and selective, competitive antagonist of TRPV1.
M6373 A 784168 A 784168 is a potent and selective TRPV1 antagonist.
M6250 AM-0902 AM-0902 is a potent, selective antagonist of TRPA1 with IC50s of 71 and 131 nM for rTRPA1 and hTRPA1, respectively.
M5349 (+)-Camphor Camphor is a waxy, flammable, white or transparent solid with a strong aroma, often used to relieve pain, reduce itching and treat fungal infections. It can activate TRPV1 and TRPV3.
M4513 Dihydrocapsaicin Dihydrocapsaicin is a natural capsaicin that is a selective TRPV1 agonist and increases P-Akt levels. Dihydrocapsaicin can enhance hypothermic induced neuroprotection.
M4122 8-Gingerol 8-gingerol is derived from the rhizome of ginger (Z. officinale). It has oral activity and can activate TRPV1 with EC50 of 5.0 µM. 8-Gingerol inhibited COX-2 and h. pylori growth in vitro.
M3187 Optovin Optovin is a reversible photoactivated TRPA1 activator. Optovin activates TRPA1 via structure-dependent photochemical reactions with redox-sensitive cysteine residues.
M2934 Phenazopyridine hydrochloride Phenazopyridine HCl is a competitive SARM1 inhibitor as well as a TRPM8 antagonist with an IC50 for SARM1 inhibition of 145 μM. It has local anesthetic/analgesic activity and can be used in studies related to traumatic brain injury, peripheral neuropathy, and neurodegenerative diseases.
M2591 Icilin Icilin is a synthetic super-agonist of the transient receptor potential M8 (TRPM8) ion channel.
M2383 AMG-517 AMG 517 is a potent and selective TRPV1 antagonist, antagonizes capsaicin, proton, and heat activation of TRPV1 with IC50 of 0.76 nM, 0.62 nM and 1.3 nM.
M2087 HC-030031 HC-030031 is a selective TRPA1 blocker, antagonizing TRPA1-mediated calcium influx induced by AITC and formalin (IC50 = 6.2 and 5.3 μM, respectively).
M1846 SB-705498 SB-705498 is a potent, selective and orally bioavailable transient receptor potential vanilloid 1 (TRPV1) receptor antagonist with a pIC50 of 7.1.
M52704 N-Oleoyl glutamine N-oleoyl-glutamine is a PM20D1-regulated N-acyl amino acids (NAAs).

Products are for research use only. Not for human use. We do not sell to patients.
© Copyright 2010-2023 AbMole BioScience. All Rights Reserved.