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Probenecid

Cat. No. M2960

All AbMole products are for research use only, cannot be used for human consumption.

Probenecid  Structure
Synonym:

Benemid

Size Price Availability Quantity
Free Sample (0.5-1 mg)  USD 0 In stock
10mM*1mL in DMSO USD 50  USD50 In stock
500mg USD 40  USD40 In stock
1g USD 55  USD55 In stock
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Quality Control & Documentation
Biological Activity

Probenecid is a classical competitive inhibitor of organic anion transport, which is also a TRPV2 agonist and an inhibitor of TAS2R16.

Product Citations
Chemical Information
Molecular Weight 285.36
Formula C13H19NO4S
CAS Number 57-66-9
Solubility (25°C) DMSO 47 mg/mL
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Richard J Everts, et al. Probenecid effects on cephalexin pharmacokinetics and pharmacodynamics in healthy volunteers

[2] Richard J Everts, et al. Probenecid and food effects on flucloxacillin pharmacokinetics and pharmacodynamics in healthy volunteers

[3] Ana Laura Coln-Gonzlez, et al. Probenecid: an emerging tool for neuroprotection

[4] Nathan Robbins, et al. The history and future of probenecid

[5] G R Brown. Cephalosporin-probenecid drug interactions

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Keywords: Probenecid , Benemid supplier, TRP Channel, inhibitors, activators

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