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5-HT Receptor 5-hydroxytryptamine receptor

Cat.No.  Name Information
M2048 Sumatriptan succinate Sumatriptan succinate (GR 43175) is an orally active 5-HT1 receptor agonist with Kis of 17 nM, 27 nM and 100 nM for 5-HT1D, 5-HT1B and 5-HT1A receptors, respectively. Sumatriptan succinate can be used for the research of migraine headache.
M3417 Clozapine Clozapine is a potent 5-HT1C receptor antagonist with an IC50 of 110 nM for 5-HT-stimulated phosphoinositide hydrolysis.
M2821 Lorcaserin hydrochloride Lorcaserin hydrochloride is a selective full agonist of human 5-HT2C receptor with Ki of 15 nM.
M5656 Fluoxetine hydrochloride Fluoxetine hydrochloride is an antidepressant of the selective serotonin reuptake inhibitor (SSRI) class.
M14577 Fluoxetine Fluoxetine (LY-110140 free base) is a selective serotonin reuptake inhibitor (SSRI) class used for antidepressant research.
M3659 Pimavanserin Pimavanserin is a selective serotonin 5-HT2A inverse agonist, with pIC50 and pKd of 8.73 and 9.3, respectively.
M3006 Sertraline hydrochloride Sertraline hydrochloride is a 5-HT antagonist with Ki of 13 nM.
M56085 LY334370 hydrochloride  LY334370 hydrochloride is a selective 5-HT1F receptor agonist with a Kd value of 0.446 nM.
M56084 SB 243213 hydrochloride  SB 243213 hydrochloride is an orally active, selective and high-affinity 5-HT2C receptor antagonist with a pKi of 9.37 and a pKb of 9.8 for human 5-HT2C receptor.
M56083 SB-224289 hydrochloride SB-224289 hydrochloride is a selective 5-HT1B receptor antagonist, with anxiolytic effect.
M56082 LY 344864 hydrochloride  LY 344864 hydrochloride is a selective, orally active 5-HT1F receptor agonist with a Ki of 6 nM.
M56081 SB 258719 hydrochloride  SB 258719 hydrochloride is a selective 5-HT7 receptor antagonist displayed high affnity (pKi=7.5) for the receptor.
M56080 Zacopride hydrochloride  Zacopride hydrochloride is a highly potent 5-HT3 receptor antagonist with Kis of 0.38 and 373 nM for 5-HT3 and 5-HT4 receptor, respectively.
M56079 Anpirtoline hydrochloride Anpirtoline hydrochloride is a hydrochloride of anpirtoline.
M56078 SB 243213 dihydrochloride  SB 243213 dihydrochloride is an orally active, selective and high-affinity 5-HT2C receptor antagonist with a pKi of 9.37 and a pKb of 9.8 for human 5-HT2C receptor.
M56077 (R)-Viloxazine hydrochloride  (R)-Viloxazine hydrochloride is a less active R-isomer of Viloxazine hydrochloride.
M56076 Tedatioxetine hydrobromide Tedatioxetine (Lu AA24530) hydrobromide acts as a serotonin and norepinephrine (NE)-preferring triple reuptake inhibitor (TRI) and 5-HT2A, 5-HT2C, 5-HT3 and α1A-adrenergic receptor antagonist.
M56075 R(+)-8-OH-DPAT hydrobromide R(+)-8-OH-DPAT ((R)-8-Hydroxy-2-dipropylaminotetralin) hydrobromide is a potent 5-HT1A agonist.
M56074 NPS ALX Compound 4a dihydrochloride  NPS ALX Compound 4a dihydrochloride is a potent and selective 5-hydroxytryptamine6 (5-HT6) receptor antagonist, with an IC50 of 7.2 nM and a Ki of 0.2 nM.
M54819 TC-2153 TC-2153 is a selective inhibitor of striatal-enriched protein tyrosine phosphatase (STEP). TC-2153 also inhibits 5-HT2A receptor-mediated signaling.
M54777 Gentisein Gentisein (NSC-329491), the major metabolite of Mangiferin, shows the most potent serotonin uptake inhibition with an IC50 value of 4.7 µM.
M54692 MM120 MM120 is a synthetic tryptamine that is also a partial agonist at the 5-hydroxytryptamine 2A (5-HT2A) receptor. It can be used in studies related to GAD and attention deficit hyperactivity disorder (ADHD).
M54596 SB 258741 hydrochloride SB 258741 hydrochloride is a specific 5-HT7 receptor antagonist for schizophrenia.
M54595 5-HT1A antagonist 1 5-HT1A antagonist 1 is a potent and selective 5-HT1A receptor antagonist with a Ki value of 35 nM.5-HT1A antagonist 1 can be used in the study of central nervous system disorders.
M54513 Nemifitide diTFA Nemifitide diTFA (INN 00835 diTFA) is a synthetic pentapeptide antidepressant with a potential for rapid onset of action.
M53845 4-Chloro-L-phenylalanine 4-Chloro-L-phenylalanine (L-PCPA) is a 5-HT biosynthesis inhibitor.
M53286 CART(62-76)(human, rat) CART(62-76)(human,rat) is a neuropeptide (62-76 residues of the CART peptide) with neurotransmitter-like effects.




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