| Cat.No. | Name | Information |
|---|---|---|
| M4973 | BAPTA-AM | BAPTA-AM is a selective, membrane-permeable calcium chelator. BAPTA-AM inhibits hERG channels, hKv1.3 and hKv1.5 channels in HEK 293 cells with IC50s of 1.3 μM, 1.45 μM and 1.23 μM, respectively. |
| M2181 | ML133 hydrochloride | ML133 hydrochloride is a selective inhibitor of the Kir2 family of inward rectifier (IRK, KCNJ) potassium channels. |
| M3456 | Chlorpromazine hydrochloride | Chlorpromazine hydrochloride is an antagonist of D2, 5HT2A, potassium and sodium channels. The Ki of Chlorpromazine Hydrochloride to D2 and 5HT2A were 363 nM and 8.3 nM, respectively. Chlorpromazine also excites the 20S proteasome. *The compound is unstable in solutions, freshly prepared is recommended |
| M7029 | Nigericin sodium salt | Nigericin (NSC 292567) sodium salt is a selective K+ ionophore, Nigericin sodium salt is also an NLRP3 activator which can activate NLRP3 inflammasome to induce pro-inflammatory and immunostimulatory processes. |
| M20428 | Retigabine 2HCl | Retigabine is a novel anticonvulsant with activity in a broad range of seizure models. The mechanism of action involves opening of neuronal K(V)7.2-7.5 (formerly KCNQ2-5) voltage-activated K(+) channels. |
| M9780 | Nigericin | Nigericin is an antibiotic derived from Streptomyces hygroscopicus, it acts as an H+, K+, Pb2+ ionophore. |
| M52752 | Phe-Met-Arg-Phe, amide acetate | Phe-Met-Arg-Phe, amide acetate dose dependently (ED50=23 nM) activates a K+ current in the peptidergic caudodorsal neurons. |
| M52751 | Charybdotoxin | Charybdotoxin, a 37-amino acid peptide, is a K+ channel blocker. |
| M52750 | Agitoxin-2 | Agitoxin-2 is a K+ channel inhibitor, with IC50 values of 201 pM and 144 pM for mKV1.3 and mKV1.1, respectively). |
| M52748 | OSK-1 | OSK-1 is a potent Kv channel blocker with IC50s of of 0.6 nM, 5.4 nM, 0.014 nM for Kv1.1, Kv1.2 and Kv1.3, respectively. |
| M52747 | Guangxitoxin 1E | Guangxitoxin 1E is a potent and selective blocker of KV2.1 and KV2.2 channels. |
| M52746 | κM-Conotoxin RIIIK | κM-Conotoxin RIIIK is a potassium channel antagonist. |
| M52745 | δ-Dendrotoxin | δ-Dendrotoxin is a K+ channel blocker that can be obtained from the venom of the black mamba snake. |
| M52744 | Docosahexaenoyl glycine | Docosahexaenoyl glycine is a PUFA analogue. |
| M52743 | Phe-Met-Arg-Phe, amide | Phe-Met-Arg-Phe, amide dose dependently (ED50=23 nM) activates a K+ current in the peptidergic caudodorsal neurons. |
| M52742 | Tyr-Somatostatin-28 | Tyr-Somatostatin-28 is a somatostatin that adds a Tyrosine amino acid to Somatostatin-28. |
| M52741 | β-Bag cell peptide | β-Bag cell peptide is a neuroactive peptide. |
| M52740 | Heteropodatoxin-2 | Heteropodatoxin-2, a peptides of 30-amino acid, is a heteropodatoxin. |
| M52739 | Kaliotoxin (1-37) | Kaliotoxin (1-37) is a toxin from the scorpion Artdroctonus mauretanicus mauretanicus. |
| M52738 | Pandinotoxin Kα | Pandinotoxin Kα, isolated from the venom of Pandinus imperator, is the inhibitor of A-type potassium channel. |
| M52737 | Dendrotoxin K | Dendrotoxin K is a Kv1.1 channel blocker. |
| M52736 | Dendrotoxin-I | Dendrotoxin-I is a potent K+ channels blocker and targets voltage-gated potassium channel subunits KV1.1 and KV1.2. |
| M52735 | Phrixotoxin 2 | Phrixotoxin 2 is a highly selective KV4.2 and KV4.3-channels blocker. |
| M52733 | Stromatoxin 1 | Stromatoxin 1 is an inhibitor of Potassium Channel, a peptide which can be isolated from tarantulas. |
| M52732 | Noxiustoxin | Noxiustoxin is a toxin from the venom of the Mexican scorpion Centruroides noxius which block voltage-dependent potassium channel (Kv1.3, IC50 = 360 nM), and calcium-activated potassium channel. |
| M52731 | Kaliotoxin | Kaliotoxin is a peptidyl inhibitor of neuronal BK-Type. |
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