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Aryl hydrocarbon Receptor Aryl Hydrocarbon Receptor (AhR)

Inhibitor/Activator

Cat.No.  Name Information
M8807 Perillaldehyde Perillaldehyde inhibits BaP-induced AHR activation and ROS production, inhibits BaP/AHR-mediated release of the CCL2 chemokine, and activats the NRF2/HO1 antioxidant pathway.
M7727 CH-223191 CH-223191 is a potent and specific aryl hydrocarbon receptor (AhR) antagonist. CH-223191 inhibits TCDD-mediated nuclear translocation and DNA binding of AhR, and inhibits TCDD-induced luciferase activity with an IC50 of 0.03 μM. *The compound is unstable in solutions, freshly prepared is recommended
M38970 Benzyl butyl phthalate Benzyl butyl phthalate can trigger the migration and invasion of hemangioma (HA) cells via upregulation of Zeb1. Benzyl butyl phthalate activates aryl hydrocarbon receptor (AhR) in breast cancer cells to stimulate SPHK1/S1P/S1PR3 signaling and enhances formation of metastasis-initiating breast cancer stem cells (BCSCs).
M25533 Carbidopa monohydrate Carbidopa monohydrate is a dopa decarboxylase (DDC) inhibitor, which can be used for the research of Parkinson's disease. Carbidopa monohydrate is also a selective aryl hydrocarbon receptor (AhR) modulator.
M25481 β-Naphthoflavone β-Naphthoflavone is an aryl hydrocarbon receptor (AhR) agonist, used as a positive control for the induction of AhR transcriptional activity. β-Naphthoflavone inhibits hydrogen peroxide-induced apoptosis.
M20602 UM729 UM729 is an enhancer of aryl hydrocarbon receptor (AhR) antagonists.
M11147 Skatole Skatole is a substance produced by the intestinal flora that regulates intestinal epithelial cell function by activating aryl hydrocarbon receptors and p38.
M10941 Tapinarof Tapinarof (WBI-1001) is a Frist in class aromatic hydrocarbon receptor (AhR) agonist with EC50 of 13 nM. Tapinarof reduced skin inflammation in mice. It can effectively inhibit inflammatory cytokines, regulate skin barrier protein expression and antioxidant activity.
M10486 GNF351 GNF351 is a full aryl hydrocarbon receptor (AHR) antagonist. GNF351 competes with a photoaffinity AHR ligand for binding to the AHR with an IC50 of 62 nM.
M10243 D-Kynurenine D-kynurenine is a metabolite of D-tryptophan, which can be used as a biological precursor of KYNA and 3-hydroxykynurenine.
M9723 L-Kynurenine L-Kynurenine is an aryl hydrocarbon receptor agonist.
M9714 CAY10465 CAY10465 is an analog of resveratrol acting as a potent and selective aryl hydrocarbon receptor agonist, with a Ki of 0.2 nM.
M9693 PDM2 PDM2 is a potent and selective aryl hydrocarbon receptor (AhR) antagonist, with a Ki of 1.2 nM.
M9490 YL-109 YL-109 is a novel anticancer agent, which can inhibit breast cancer cell growth and invasiveness in vitro and in vivo, YL-109 is also an STUB1 enhancer.
M9087 FICZ FICZ is a potent aryl hydrogen receptor (AhR) agonist.
M8862 YH439 YH439 is an aryl hydrocarbon receptor activator.
M4783 Diosimin Diosimin is a flavonoid glycoside found in citrus fruits, hyssop, and rosemary.
M3260 Carbidopa Carbidopa is an aromatic-L-amino-acid decarboxylase inhibitor with an IC50 of 29 ± 2 μM.
M2577 StemRegenin 1 StemRegenin 1 is an AhR inhibitor with IC50 of 127 nM.
M41957 KYN-101 KYN-101 is a potent, selective and orally active AHR inhibitor.




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