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Cat.No.	Name	Information
M2206	TH-302 (Evofosfamide)	TH-302 is a highly potent and selective hypoxia-activated procompound targeting hypoxic regions of solid tumors with IC50 of 19 nM.
M6098	Baicalein	Baicalein is a CYP2C9 and prolyl endopeptidase inhibitor, IC50 value of 3.12 mM.
M9325	EGTA	EGTA is a specific calcium chelator with a Kd of 60.5 nM at physiological pH (7.4) and a high specificity for Ca2+ than for Mg2+.EGTA significantly inhibits the substrate adhesion capacity of inflammatory macrophages.
M9330	Brij-35	Brij-35 (Polidocanol) is a high HLB, ethoxylated, nonionic ether of lauryl alcohol with broad pH stability.
M6154	2-PMPA tetrasodium	2-PMPA (PMPA tetrasodium salt) is a potent and selective inhibitor of glutamate carboxypeptidase II (GCPII) with an IC50 of 300 pM.
M2250	Pamidronate disodium	Pamidronate disodium is a nitrogen containing bisphosphonate, used to the research of preventing osteoporosis.
M9916	DPPH	DPPH (2,2-Diphenyl-1-picrylhydrazyl) is a stable free radical that measures the free radical scavenging activity of antioxidants.
M9194	Insulin (human)	Insulin (human) is a polypeptide hormone that regulates the level of sugar (glucose) in the blood and is produced by beta cells of islets.
M3409	Formestane	Formestane is a second generation selective aromatase inhibitor with an IC50 of 80 nM.
M9665	N-(2-amino-2-oxoethyl)acrylamide	N-(2-Amino-2-oxoethyl)acrylamide
M8563	Macelignan	Macelignan is a neuroprotective lingan isolated from nutmeg (Myristica fragrans) that protects dopaminergic neurons from inflammatory degeneration.
M8562	SID 3712249	SID 3712249 (MiR-544 Inhibitor 1) is an inhibitor of the biogenesis of microRNA-544 (miR-544).
M8559	SR1848	SR1848 is a cell penetrant and potent inhibitor of orphan nuclear receptor liver receptor homolog 1 (LRH-1; NR5A2) that reduces the expression of CyclinD1 and E1, which results in inhibition of cell proliferation.
M8557	CS1	CS1 is a selective and potent inhibitor of topoisomerase IIα (TopoIIα) that potently inhibits a proliferation of cancer cell lines including MDA-MB-231 and A548 cells, with less toxicity than etoposide.
M8556	KY-05009	KY-05009 is a Traf2- and Nck-interacting kinase (TNIK) inhibitor that inhibits the epithelial-to-mesenchymal transition (EMT) in cancer cells.
M8554	LW479	LW479 is a potent histone deacetylase inhibitor (HDACI) that down-regulates EGFR expression.
M8553	ABT-089 dihydrochloride	ABT-089 (Pozanicline) is a subtype-selective neuronal nicotinic receptor partial agonist binding primarily to the α4β2 and also α6β2 subtypes.
M8552	Allyphenyline oxalate	Allyphenyline is a potent α2C-adrenoceptor/serotonin 5-HT1A receptor agonist and α2A-adrenoceptor antagonist that exhibits anxiolytic effect and antidepressant activity.
M8551	Ogerin negative control	Ogerin negative control is a structurally similar analog of ogerin (catalog no.
M8550	Ogerin	Ogerin is a selective positive allosteric modulator of an orphan GPCR, GPR68, also known as Ovarian cancer G-protein coupled receptor 1 (OGR1).
M8549	FzM1	FzM1 is an allosteric ligand of the Frizzled4 (Fz4) receptor and a Wnt/β-catenin pathway inhibitor, found by a screen for pharmacological chaperones for a misfolded mutant of the Frizzled4 (Fz4) receptor.
M8548	Ophiobolin A	Ophiobolin A is a fungal metabolite, toxic to many crops and found to have antimicrobial and anticancer activity.
M8547	Thiocolchicoside	Thiocolchicoside is a potent competitive γ-aminobutyric acid type A (GABAA) receptor antagonist and glycine receptor agonist with muscle relaxant, anti-inflammatory, and analgesic activity.
M8546	Chlorcyclizine	Chlorocyclozine is a first-generation antihistamine compound that is being investigated as a potential hepatitis C agent.
M8544	ABH hydrochloride	ABH (2(S)-amino-6-boronohexanoic acid) is a highly potent and specific arginase inhibitor that inhibits the LPS-induced increases in pulmonary IL-8, neutrophils and goblet cells as well as airway fibrosis in rodent model of COPD.
M8542	Practolol	Practolol is a potent and selective β-adrenoceptor antagonist.
M8540	Ibufenac	Ibufenac is a non-steroidal anti-inflammatory drug (NSAID) analog of ibuprofen that was withdrawn for hepatotoxicity.
M8539	G3335	G3335 ( L-tryptophyl-L-glutamic acid) is a cell-permeable dipeptide that acts as a selective and reversible PPARγ antagonist with a Kd value of 8.
M8537	KS 370G	KS370G is a synthetic caffeamide derivative that exhibits hypoglycemic effects in mice model of diabetes.
M8534	Ac-YVAD-pNA	Ac-YVAD-pNA is a very selective chromogenic substrate for caspase-1, a key mediator of inflammatory processes formerly known as interleukin (IL)-1-converting enzyme.

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