| Cat.No. | Name | Information |
|---|---|---|
| M2206 | TH-302 (Evofosfamide) | TH-302 is a highly potent and selective hypoxia-activated procompound targeting hypoxic regions of solid tumors with IC50 of 19 nM. |
| M6098 | Baicalein | Baicalein is a CYP2C9 and prolyl endopeptidase inhibitor, IC50 value of 3.12 mM. |
| M9325 | EGTA | EGTA is a specific calcium chelator with a Kd of 60.5 nM at physiological pH (7.4) and a high specificity for Ca2+ than for Mg2+.EGTA significantly inhibits the substrate adhesion capacity of inflammatory macrophages. |
| M9330 | Brij-35 | Brij-35 (Polidocanol) is a high HLB, ethoxylated, nonionic ether of lauryl alcohol with broad pH stability. |
| M6154 | 2-PMPA tetrasodium | 2-PMPA (PMPA tetrasodium salt) is a potent and selective inhibitor of glutamate carboxypeptidase II (GCPII) with an IC50 of 300 pM. |
| M2250 | Pamidronate disodium | Pamidronate disodium is a nitrogen containing bisphosphonate, used to the research of preventing osteoporosis. |
| M9916 | DPPH | DPPH (2,2-Diphenyl-1-picrylhydrazyl) is a stable free radical that measures the free radical scavenging activity of antioxidants. |
| M9194 | Insulin (human) | Insulin (human) is a polypeptide hormone that regulates the level of sugar (glucose) in the blood and is produced by beta cells of islets. |
| M3409 | Formestane | Formestane is a second generation selective aromatase inhibitor with an IC50 of 80 nM. |
| M9665 | N-(2-amino-2-oxoethyl)acrylamide | N-(2-Amino-2-oxoethyl)acrylamide |
| M8796 | TCPOBOP | TCPOBOP enhances the nuclear receptor CAR transactivation of cytochrome P450 (CYP), as dose-dependent direct agonist of CAR. |
| M8795 | Thioperamide maleate salt | Potent and selective H3 histamine receptor antagonist that crosses the blood-brain barrier. |
| M8794 | Trifluperidol hydrochloride | Trifluperidol hydrochloride is a dopamine receptor antagonist with antipsychotic effects and has been used in studies of schizophrenia. |
| M8793 | Tocainide hydrochloride | Tocainide hydrochloride is a sodium channel blocker; Class IB antiarrhythmic. |
| M8792 | TD52 | TD52, an erlotinib analog, is a putative inhibitor of CIP2A that exhibits potent antitumor efficacy on HCC and TNBC cells. |
| M8791 | TB5 | TB5 is a potent and selective reversible inhibitor of monoamine oxidase B (MAOB) with a Ki value of 110 nM. |
| M8790 | MDL-860 | MDL-860 is a 5-nitro-2-phenoxybenzonit |
| M8786 | Roflupram | Roflupram (FFPM) is a potent anti-inflammatory phosphodiesterase 4 (PDE4) inhibitor that was found to suppress inflammasome activation in microglial cells by enhancing autophagy. |
| M8785 | Fosamprenavir calcium | Fosamprenavir calcium is an HIV protease inhibitor anti-retroviral. |
| M8782 | NAMI-A | NAMI-A is a potent antimetastatic compound in vivo that is exhibits little cytotoxicity towards many cancer cell lines. |
| M8778 | ZD0947 | ZD0947 is potent ATP-sensitive K+ channels (KATP channels) opener. |
| M8777 | BPAM344 | BPAM344 is a potent positive allosteric modulator (PAM) on the three KAR subunits GluK1b, GluK2a, and GluK3a. |
| M8776 | ARM390 | ARM390 in a δ-selective opioid receptor agonist derivative of SNC80. |
| M8775 | DMAT | Casein kinase II inhibitor II (Ck2 Inhibitor II) is a high affinity ATP-competitive inhibitor of casein kinase II. |
| M8773 | Liarozole dihydrochloride | Liarozole (R 75251, R75,251) is an orally active benzimidazole-based retinoic acid (RA) metabolism blocking agent (RAMBA) that targets multiple P450 enzymes, including aromatase (CYP19), 17-hydroxylase/17,20-lyas |
| M8772 | SAK3 | SAK3 is a potent and orally active spiroimidazopyridine derivative that enhances Cav3. |
| M8771 | SR2595 | SR2595 is an inverse agonist of PPARG (PPARγ) with an IC50 value of 30 nM. |
| M8770 | Didox | Didox is a ribonucleotide reductase (RNR) inhibitor that inhibits proliferation of and decreased secretion of cytokines IL-6, IFN-g, TNF-a, IL-2, IL-13, IL-10 and IL-4. |
| M8768 | TUG-1387 | TUG-1387 is a close structural analog of AH-7614 that lacks activity at FFA4 that can serve as negative control. |
| M8767 | MIND4-17 | MIND4-17 is a potent NRF2 (nuclear factor erythroid 2-related factor 2) activator that covalently modifies a critical stress-sensor cysteine (C151) in the BTB domain of the E3 ligase substrate adaptor protein Kelch-like ECH-associated protein 1 (KEAP1), the primary negative regulator of NRF2. |
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