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Abmole Inhibitor Catalog 2017

Estrogen Receptor Estrogen Receptor


Cat.No.  Name Information
M10348 27-Hydroxycholesterol 27-Hydroxycholesterol is a selective estrogen receptor modulator, and it is also an agonist of the liver X receptor.
M10254 SAR439859 (Amcenestrant) SAR439859 (Amcenestrant) is an orally active, nonsteroidal and selective degrader of estrogen receptor, it is also a potent antagonist of ER with EC50 of 0.2 nM for ERα degradation.
M10252 4-Hydroxytamoxifen 4-Hydroxytamoxifen is a selective estrogen receptor modulator.
M9967 Methylpiperidino pyrazole Methylpiperidino pyrazole (MPP) is an agonist for estrogen receptor α and lacks any ligand functionality with estrogen receptor (ER)β.
M9796 Endoxifen E-isomer hydrochloride Endoxifen E-isomer hydrochloride is a tamoxifen metabolite and potent Selective Estrogen Response Modifier (SERM).
M9197 Relugolix Relugolix, also known as TAK-385, is a luteinizing hormone-releasing hormone (LH-RH) receptor antagonist with an IC50 of 0.12 nM.
M9196 Elagolix sodium Elagolix Soidum is a potent, selective, orally active, non-peptide antagonist of the gonadotropin-releasing hormone receptor (GnRHR) with Kd value of 54 pM.
M8953 GDC-0810 GDC-0810 (Brilanestrant, ARN-81) is an orally bioavailable selective estrogen receptor degrader (SERD) with IC50 of 0.7 nM.
M8508 PHTPP PHTPP is a selective estrogen receptor β (ERβ) full antagonist with 36-fold selectivity for ERβ over ERα.
M7871 G15 G15 is a high affinity and selective G-protein-coupled estrogen receptor (GPER/GPR30) antagonist with a Ki of 20 nM.
M7839 (E/Z)-4-Hydroxytamoxifen Metabolite of the chemotherapeutic drug tamoxifen, exhibiting more potent estrogen agonist/antagonist activity than the parent drug.
M7353 Tamoxifen Tamoxifen is a estrogen receptor partial agonist/antagonist.
M6710 Endoxifen hydrochloride Endoxifen hydrochloride is a potent antiestrogen; ERα ligand.
M6165 GSK 4716 GSK 4716 is a selective agonist with estrogen-related receptors ERRβ and ERRγ.
M5917 Raloxifene HCl RaloxifeneHcl(LY156758 Hcl) is a second generation selective estrogen receptor antagonist.
M5902 Progesterone Progesterone is an endogenous steroid hormone involved in the menstrual cycle, pregnancy, and embryogenesis of humans and other species. A potent agonist of the nuclear progesterone receptor (nPR) with Kd of 1 nM; An agonist of the membrane progesterone receptors(mPRs); An antagonist of the σ1 receptor.
M5765 Megestrol Acetate Megestrol acetate is a synthetic progestogen, used to treat breast cancer and loss of appetite.
M5764 Medroxyprogesterone acetate Medroxyprogesterone acetate (MPA) is a synthetic progestin and act as a potent progesterone receptor agonist, used to treat abnormal menstruation or irregular vaginal bleeding.
M5735 Leuprolide Acetate Leuprolide acetate (Leuprorelin) is a GnRH analog; leuprolide acetate acts as an agonist at pituitary GnRH receptors.
M5698 Hydroxyprogesterone caproate Hydroxyprogesterone Caproate is a synthetic progestational agent. It binds to and activates nuclear progesterone receptors in the reproductive system and inhibits ovulation and an alteration in the cervical mucus and endometrium.
M5668 Bavachin Bavachin, a flavonoid first isolated from seeds of P. corylifolia, acts as a phytoestrogen that activates the estrogen receptors ERα and ERβ with EC50s of 320 and 680 nM, respectively.
M5635 Etonogestrel Etonogestrel is a synthetic form of the naturally occurring female sex hormone progesterone. It binds to the cytoplasmic progesterone receptors in the reproductive system and subsequently activates progesterone receptor mediated gene expression.
M5628 Ethisterone Ethisterone is a progestogen hormone being considered to treat prostate cancer.
M5627 Estropipate Estropipate is a form of estrogen, used to treat symptoms of menopause, also used to prevent osteoporosis.
M5625 Estradiol Estradiol (17β-estradiol) is a human sex hormone and steroid, and the primary female sex hormone.
M5599 Drospirenone Drospirenone is a synthetic progestin that is an analog to spironolactone.
M5564 Desogestrel Desogestrel is a synthetic progestational hormone used often as the progestogenic component of combined oral contraceptive agents.
M5511 Chlormadinone acetate Chlormadinone acetate is a steroidal progestin with additional antiandrogen and antigonadotropic effects, used often in combinations as an oral contraceptive. Its half-life is about 34-38 hours.
M4836 G-1 G-1 is a potent and selective GPR30 receptor agonist (Ki = 11 nM, EC50 = 2 nM).
M4835 DPN DPN is a highly potent estrogen ERβ receptor agonist with a 70-fold selectivity over ERα with EC50 values are 0.85 and 66 nM,respectively.
M4834 PPT PPT is a potent subtype-selective estrogen receptor agonist with EC50 ~ 200 pM and displays 410-fold selectivity for ERα over ERβ.
M4368 Kaempferol Kaempferol is a natural flavonol, functions as an ERRα and ERRγ inverse agonist.
M3945 Estrone Estrone is an estrogenic hormone.
M3764 DY131 DY131(GSK 9089) is a novel selective agonist of ERRβ and ERRγ which displays minimal activity at ERRα, ERα and ERβ at concentrations up to 30 μM.
M3692 Chlorotrianisene Chlorotrianisene is a therapeutic estrogen which inhibits bone loss and delay the atrophy of uterus.
M3652 Ospemifene Ospemifene is a non-hormonal selective estrogen receptor modulator (SERM) which is used for the treatment of dyspareunia.
M3580 L-carnitine L-carnitine is constituent of striated muscle and liver. It is used therapeutically to stimulate gastric and pancreatic secretions and in the treatment of hyperlipoproteinemias.
M3564 Clomifene citrate Clomifene citrate is a selective estrogen receptor modulator.
M3392 Ethinyl Estradiol Ethinyl Estradiol is an orally bio-active estrogen used in almost all modern formulations of combined oral contraceptive pills.
M3371 Estriol Estriol is an antagonist of the G-protein coupled estrogen receptor in estrogen receptor-negative breast cancer cells.
M3333 Hexestrol Hexestrol binds to ERα and ERβ with EC50 of 0.07 nM and 0.175 nM, respectively.
M2683 Estradiol Benzoate Estradiol benzoate is an estradiol analog which binds to the human, murine and chicken ERα with IC50 of 22-28 nM.
M2516 Cholesterol Cholesterol is the principal sterol of all higher animals required to build and maintain membranes.
M2280 Tamoxifen Citrate (ICI 46474) Tamoxifen Citrate is an antagonist of the estrogen receptor by competitive inhibition of estrogen binding.
M2174 Calcitriol Calcitriol is an Active metabolite of vitamin D3 that activates the vitamin D receptor.
M2097 LY500307 LY500307 is a potent, selective estrogen receptor beta agonist with an EC50 of 0.66 nM.
M1966 Fulvestrant Fulvestrant (Faslodex) is a novel estrogen receptor (ER) antagonist (IC50 = 0.29 nM).

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