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Estrogen Receptor Estrogen Receptor


Cat.No.  Name Information
M1966 Fulvestrant Fulvestrant is a Estrogen receptor (ER) antagonist with IC50 of 0.094 nM. Fulvestrant can also induce autophagy and apoptosis, and has anti-tumor effect.
M3371 Estriol Estriol is an antagonist of the G-protein coupled estrogen receptor in estrogen receptor-negative breast cancer cells.
M4368 Kaempferol Kaempferol is a natural flavonol, functions as an ERRα and ERRγ inverse agonist.
M7353 Tamoxifen Tamoxifen is a estrogen receptor partial agonist/antagonist.
M7871 G15 G15 is a high affinity and selective G-protein-coupled estrogen receptor (GPER/GPR30) antagonist with a Ki of 20 nM.
M11047 Quinestrol Quinestrol is a synthetic estrogen that has the potential to be used in breast and prostate cancer related research.
M10923 Giredestrant Giredestrant (GDC-9545) is a potential "best-in-class" selective estrogen receptor inhibitor (SERD). Giredestrant can competitively bind with Estradiol in the ER ligand binding domain and induce conformational changes. Giredestrant has antitumor activity.
M10910 Zuclomiphene citrate Zuclomiphene citrate is a cis isomer of clomiphene citrate. Zuclomiphene citrate has an anti-estrogen effect and inhibits the secretion of luteinizing hormone (LH) more than trans isomers. Zuclomiphene citrate is also an oral active cholesterol lowering agent.
M10348 27-Hydroxycholesterol 27-Hydroxycholesterol is a selective estrogen receptor modulator, and it is also an agonist of the liver X receptor.
M10254 SAR439859 (Amcenestrant) SAR439859 (Amcenestrant) is an orally active, nonsteroidal and selective degrader of estrogen receptor, it is also a potent antagonist of ER with EC50 of 0.2 nM for ERα degradation.
M10252 4-Hydroxytamoxifen 4-Hydroxytamoxifen is a selective estrogen receptor modulator.
M9967 Methylpiperidino pyrazole Methylpiperidino pyrazole (MPP) is an agonist for estrogen receptor α and lacks any ligand functionality with estrogen receptor (ER)β.
M9796 Endoxifen E-isomer hydrochloride Endoxifen E-isomer hydrochloride is a tamoxifen metabolite and potent Selective Estrogen Response Modifier (SERM).
M9197 Relugolix Relugolix, also known as TAK-385, is a luteinizing hormone-releasing hormone (LH-RH) receptor antagonist with an IC50 of 0.12 nM.
M9196 Elagolix sodium Elagolix Soidum is a potent, selective, orally active, non-peptide antagonist of the gonadotropin-releasing hormone receptor (GnRHR) with Kd value of 54 pM.
M8953 GDC-0810 GDC-0810 (Brilanestrant, ARN-81) is an orally bioavailable selective estrogen receptor degrader (SERD) with IC50 of 0.7 nM.
M8508 PHTPP PHTPP is a selective estrogen receptor β (ERβ) full antagonist with 36-fold selectivity for ERβ over ERα.
M7871 G15 G15 is a high affinity and selective G-protein-coupled estrogen receptor (GPER/GPR30) antagonist with a Ki of 20 nM.
M7839 (E/Z)-4-Hydroxytamoxifen Metabolite of the chemotherapeutic drug tamoxifen, exhibiting more potent estrogen agonist/antagonist activity than the parent drug.
M7353 Tamoxifen Tamoxifen is a estrogen receptor partial agonist/antagonist.
M6710 Endoxifen hydrochloride Endoxifen hydrochloride is a potent antiestrogen; ERα ligand.
M6165 GSK 4716 GSK 4716 is a selective agonist with estrogen-related receptors ERRβ and ERRγ.
M5917 Raloxifene HCl RaloxifeneHcl(LY156758 Hcl) is a second generation selective estrogen receptor antagonist.
M5902 Progesterone Progesterone is an endogenous steroid hormone involved in the menstrual cycle, pregnancy, and embryogenesis of humans and other species. A potent agonist of the nuclear progesterone receptor (nPR) with Kd of 1 nM; An agonist of the membrane progesterone receptors(mPRs); An antagonist of the σ1 receptor.
M5765 Megestrol Acetate Megestrol acetate is a synthetic progestogen, used to treat breast cancer and loss of appetite.

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