| Cat.No. | Name | Information |
|---|---|---|
| M1966 | Fulvestrant | Fulvestrant is a Estrogen receptor (ER) antagonist with IC50 of 0.094 nM. Fulvestrant can also induce autophagy and apoptosis, and has anti-tumor effect. |
| M3371 | Estriol | Estriol is an antagonist of the G-protein coupled estrogen receptor in estrogen receptor-negative breast cancer cells. |
| M4368 | Kaempferol | Kaempferol is an inverse agonist of ERRα and ERRγ that inhibits estrogen receptor (ER α) expression in breast cancer cells and induces apoptosis by activating MEK-MAPK in glioblastoma cells and lung cancer cells. It can be used in breast cancer research. |
| M7353 | Tamoxifen | Tamoxifen is an orally active, selective estrogen receptor partial agonist/antagonist. Tamoxifen is a potent Hsp90 activator and enhances the Hsp90 molecular chaperone ATPase activity. Tamoxifen also potent inhibits infectious EBOV Zaire and Marburg (MARV) with IC50 of 0.1 µM and 1.8 µM, respectively. |
| M7871 | G15 | G15 is a high affinity and selective G-protein-coupled estrogen receptor (GPER/GPR30) antagonist with a Ki of 20 nM. |
| M4374 | Gypenoside-XVII | Gypenoside XVII is a novel phytoestrogens belonging to gypenosides, which can activate estrogen receptors. |
| M2174 | Calcitriol | Calcitriol is an Active metabolite of vitamin D3 that activates the vitamin D receptor. *The compound is unstable in solutions, freshly prepared is recommended |
| M5625 | Estradiol | Estradiol (17β-estradiol) is a human sex hormone and steroid, and the primary female sex hormone. Estradiol can up-regulate the expression of neural markers of human endometrial stem cells (hEnSCs) and promote their neural differentiation. Estradiol (17β-estradiol) can be used to construct animal models of chronic non-bacterial prostatitis. |
| M4836 | G-1 | G-1 is a potent and selective GPR30 receptor agonist (Ki = 11 nM, EC50 = 2 nM). |
| M8508 | PHTPP | PHTPP is a selective estrogen receptor β (ERβ) full antagonist with 36-fold selectivity for ERβ over ERα. |
| M5668 | Bavachin | Bavachin, a flavonoid first isolated from seeds of P. corylifolia, acts as a phytoestrogen that activates the estrogen receptors ERα and ERβ with EC50s of 320 and 680 nM, respectively. |
| M5635 | Etonogestrel | Etonogestrel is a synthetic form of the naturally occurring female sex hormone progesterone. It binds to the cytoplasmic progesterone receptors in the reproductive system and subsequently activates progesterone receptor mediated gene expression. |
| M5628 | Ethisterone | Ethisterone is a progestogen hormone being considered to treat prostate cancer. |
| M5627 | Estropipate | Estropipate is a form of estrogen, used to treat symptoms of menopause, also used to prevent osteoporosis. |
| M5599 | Drospirenone | Drospirenone is a synthetic progestin that is an analog to spironolactone. |
| M5564 | Desogestrel | Desogestrel is a synthetic progestational hormone used often as the progestogenic component of combined oral contraceptive agents. |
| M5511 | Chlormadinone acetate | Chlormadinone acetate is a steroidal progestin with additional antiandrogen and antigonadotropic effects, used often in combinations as an oral contraceptive. Its half-life is about 34-38 hours. |
| M5434 | Avobenzone | Avobenzone is an oil soluble ingredient used in sunscreen products to absorb the full spectrum of UVA rays and a dibenzoylmethane derivative. |
| M4835 | DPN | DPN is a highly potent estrogen ERβ receptor agonist with a 70-fold selectivity over ERα with EC50 values are 0.85 and 66 nM,respectively. |
| M4834 | Propyl pyrazole triol (PPT) | PPT is a potent subtype-selective estrogen receptor agonist with EC50 ~ 200 pM and displays 410-fold selectivity for ERα over ERβ. |
| M4512 | Tectoridin | Tectoridin is an isoflavone isolated from Maackia Amurensis. Tectoridin is a phytoestrogen that activates estrogen and thyroid hormone receptors. Tectoridin exerts estrogenic effects through the ER dependent genomic pathway and the GPR30 dependent non-genomic pathway. |
| M4369 | Kaempferide | Kaempferide is an O-methylated flavonol also found in kaempferia galanga. Kaempferide has antiviral activity. |
| M4008 | Liquiritigenin | Liquiritigenin, a flavanone isolated from Glycyrrhiza uralensis, is a highly selective estrogen receptor β (ERβ) agonist with an EC50 of 36.5 nM for activation of the ERE tk-Luc. |
| M3945 | Estrone | Estrone is an estrogenic hormone. |
| M3764 | DY131 | DY131(GSK 9089) is a novel selective agonist of ERRβ and ERRγ which displays minimal activity at ERRα, ERα and ERβ at concentrations up to 30 μM. |
| M3692 | Chlorotrianisene | Chlorotrianisene is a therapeutic estrogen which inhibits bone loss and delay the atrophy of uterus. |
| M3652 | Ospemifene | Ospemifene is a non-hormonal selective estrogen receptor modulator (SERM) which is used for the treatment of dyspareunia. |
| M3580 | L-carnitine | L-carnitine is present in striated muscle and liver and is used in studies of hyperlipoproteinemia, stimulating gastric and pancreatic secretions. |
| M3579 | Mestranol | Mestranol is the 3-methyl ether of ethinylestradiol. It was the estrogen used in many of the first oral contraceptives. |
| M3567 | Toremifene Citrate | Toremifene Citrate is an oral selective estrogen receptor modulator (SERM) which helps oppose the actions of estrogen in the body. |
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