| Cat.No. | Name | Information |
|---|---|---|
| M1966 | Fulvestrant | Fulvestrant is a Estrogen receptor (ER) antagonist with IC50 of 0.094 nM. Fulvestrant can also induce autophagy and apoptosis, and has anti-tumor effect. |
| M3371 | Estriol | Estriol is an antagonist of the G-protein coupled estrogen receptor in estrogen receptor-negative breast cancer cells. |
| M4368 | Kaempferol | Kaempferol is an inverse agonist of ERRα and ERRγ that inhibits estrogen receptor (ER α) expression in breast cancer cells and induces apoptosis by activating MEK-MAPK in glioblastoma cells and lung cancer cells. It can be used in breast cancer research. |
| M7353 | Tamoxifen | Tamoxifen is an orally active, selective estrogen receptor partial agonist/antagonist. Tamoxifen is a potent Hsp90 activator and enhances the Hsp90 molecular chaperone ATPase activity. Tamoxifen also potent inhibits infectious EBOV Zaire and Marburg (MARV) with IC50 of 0.1 µM and 1.8 µM, respectively. |
| M7871 | G15 | G15 is a high affinity and selective G-protein-coupled estrogen receptor (GPER/GPR30) antagonist with a Ki of 20 nM. |
| M4374 | Gypenoside-XVII | Gypenoside XVII is a novel phytoestrogens belonging to gypenosides, which can activate estrogen receptors. |
| M2174 | Calcitriol | Calcitriol is an Active metabolite of vitamin D3 that activates the vitamin D receptor. *The compound is unstable in solutions, freshly prepared is recommended |
| M5625 | Estradiol | Estradiol (17β-estradiol) is a human sex hormone and steroid, and the primary female sex hormone. Estradiol can up-regulate the expression of neural markers of human endometrial stem cells (hEnSCs) and promote their neural differentiation. Estradiol (17β-estradiol) can be used to construct animal models of chronic non-bacterial prostatitis. |
| M4836 | G-1 | G-1 is a potent and selective GPR30 receptor agonist (Ki = 11 nM, EC50 = 2 nM). |
| M8508 | PHTPP | PHTPP is a selective estrogen receptor β (ERβ) full antagonist with 36-fold selectivity for ERβ over ERα. |
| M44724 | 3'-Hydroxymirificin | 3'-Hydroxymirificin is a naural compound that can be isolated from Pueraria lobata roots. |
| M43603 | ERα degrader 6 | ERα degrader 6 is an ERα degrader (KI: 75 nM). |
| M43602 | ER degrader 5 | ER degrader 5 is a potent estrogen receptor (ER) degrader. |
| M43601 | ER degrader 6 | ER degrader 6 is a potent Estrogen Receptor (ER)α degrader. |
| M43600 | Estrogen receptor modulator 7 | Estrogen receptor modulator 7 is a potent estrogen receptor modulator. |
| M43599 | ER degrader 4 | ER degrader 4 is a selective and orally active estrogen receptor degrader. |
| M43598 | SLU-PP-1072 | SLU-PP-1072 is a dual ERRα/γ inverse agonist, used in Prostate cancer (PCa) research. |
| M43597 | ERRγ agonist-2 | ERRγ agonist-2 is a potent and selective ERRγ inverse agonist with a Kd value of 6.5 μM. |
| M43596 | Yp537 TFA | Yp537 TFA is an estrogen receptor (ER) inhibitor that blocks dimerization of the human estrogen receptor. |
| M43595 | Estrogen receptor modulator 8 | Estrogen receptor modulator 8 is an orally active inhibitor of Estrogen Receptor/ERR α (IC50=0.437 nM, MCF-7 cells). |
| M43594 | Estrogen receptor antagonist 8 | Estrogen receptor antagonist 8 is a potent estrogen receptor ER antagonist with an EC50 of 4.160 μM. |
| M43593 | SLU-PP-332 | SLU-PP-332 is a pan-Estrogen Receptor/ERR agonist with EC50 values of 98, 230 and 430 nM for ERRα, ERRβ and ERRγ, respectively. |
| M43592 | ET receptor antagonist 3 | ET receptor antagonist 3 is an orally active ET receptor antagonist (IC50=0.26 nM), which can be used for research in pulmonary arterial hypertension (PAH). |
| M43591 | ET receptor antagonist 2 | ET receptor antagonist 2 is an orally active ET receptor antagonist (IC50=0.22 nM), which can be used for research in pulmonary arterial hypertension (PAH). |
| M43590 | ET receptor antagonist 1 | ET receptor antagonist 1 is an orally active ET receptor antagonist (IC50=0.18 nM), which can be used for research in pulmonary arterial hypertension (PAH). |
| M43413 | ERD-3111 | ERD-3111 is an orally active PROTAC ERα degrader (DC50: 0.5 nM). |
| M39861 | Lindleyin | Lindleyin, isolated from Rhei rhizoma, mediates hormonal effects through estrogen receptors. Lindleyin binds to ERα with estrogenic activity. |
| M39860 | Inokosterone | Inokosterone is a potential agent target of estrogen receptor 1 in rheumatoid arthritis patients. |
| M39859 | α-Zearalenol | α-Zearalenol is a Mycotoxin with high affinity for the estrogen receptors (ER), α-Zearalenol is the derivative of zearalenone (ZEN), causes reproductive disorders in animals, due to its xenoestrogenic effects. |
| M39857 | Estradiol enanthate | Estradiol enanthate is a shorter-acting estrogen. The combination of Estradiol enanthate and dihydroxyprogesterone acetophenide can be used as a monthly injectable contraceptive. |
Products are for research use only. Not for human use. We do not sell to patients.
© Copyright 2010-2024 AbMole BioScience. All Rights Reserved.
