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DPN increased GluR2 expression in the other lamina of the CA1.DPN acts as an agonist on both ER subtypes, but has a 70-fold higher relative binding affinity and 170-fold higher relative potency in transcription assays with ERbeta than with ERalpha. DPN displayed subtype-selective agonism, being ca. 30-fold more potent through ERbeta.Both PPT and DPN can acutely relax isolated mesenteric arteries with the relative potency of PPT>17beta-oestrogen>DPN.
| Molecular Weight | 239.27 |
| Formula | C15H13NO2 |
| CAS Number | 1428-67-7 |
| Solubility (25°C) | DMSO |
| Storage |
Powder -20°C 3 years ; 4°C 2 years In solvent -80°C 6 months ; -20°C 1 month |
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