Adenosine Receptor Adenosine Receptor

Inhibitors

Cat.No.	Name	Information
M4497	Norisoboldine	Norisoboldine is an isoquinoline alkaloid which acts as an AhR agonist.
M7531	AZD4635	AZD4635 is a novel adenosine 2A receptor (A2AR) inhibitor with a Ki of 1.7 nM.
M11264	KI-7	Ki-7 is an A2B adenosine receptor positive allosteric regulator. Ki-7 enhances cAMP accumulation induced by NECA, a non-selective A2B adenosine receptor agonist (EC50=445.8 nM). Ki-7 also enhanced selective A2B adenosine receptor agonist BAY 60-6583 and adenosine-induced cAMP accumulation with EC50 of 2390 nM and 2550 nM, respectively.
M10628	Adenosine amine congener	Adenosine amine congener (ADAC) is a selective A1 adenosine receptor agonist, can ameliorate noise- and cisplatin-induced cochlear injury.
M10191	Vipadenant	Vipadenant, also known as BIIB014, CEB-4520, is a potent, selective and orally available adenosine A2A receptor antagonist with Ki of 1.3 nM.
M10055	2',5'-Dideoxyadenosine	2′,5′-Dideoxyadenosine is a cell-permeable adenylyl cyclase inhibitor, IC50 = 2.7 μM in detergent-dispersed rat brain preparations.
M9888	ABT-702 dihydrochloride	ABT-702 dihydrochloride is a potent non-nucleoside adenosine kinase inhibitor, selective over other sites of adenosine interaction like A1, A2A and A3 receptors, adenosine transporter and adenosine deaminase.
M9799	Capadenoson	Capadenoson (BAY 68-4986) is an oral active, potent and selective adenosine A1 receptor agonist.
M9774	Namodenoson	Namodenoson (also known as 2-Cl-IB-MECA and CF-102) is an orally bioavailable, synthetic, highly selective adenosine A3 receptor (A3AR) agonist (Ki=0.33 nM) with potential antineoplastic activity.
M9674	MRS-3777 hemioxalate	MRS-3777 hemioxalate is a selective adenosine A3 receptor antagonist.
M9569	Etrumadenant	AB928 is an orally bioavailable, dual antagonist of the A2aR and A2bR adenosine receptors, leads to greater immunomodulatory activity and reduced tumor growth.
M7531	AZD4635	AZD4635 is a novel adenosine 2A receptor (A2AR) inhibitor with a Ki of 1.7 nM.
M7282	SCH 58261	SCH 58261 is a potent, highly selective A_2A antagonist.
M6126	CPI-444	CPI-444 is a potent and selective inhibitor of A2A receptor (A2AR) induces antitumor responses.
M5924	Regadenoson	Regadenoson is an A2A adenosine receptor agonist that is a coronary vasodilator that is commonly used in pharmacologic stress testing.
M5211	ZM241385	ZM-241385 is a high affinity antagonist ligand selective for the adenosine A2A receptor.
M4694	Theobromine	Theobromine is a methylxanthine found in cocoa beans that inhibits adenosine receptor A1 (AR1) signaling.
M4497	Norisoboldine	Norisoboldine is an isoquinoline alkaloid which acts as an AhR agonist.
M3749	Pentostatin	Pentostatin (Deoxycoformycin) is an irreversible inhibitor of adenosine deaminase (Ki = 2.5 pM).
M3228	CGS 21680	CGS 21680 is a selective adenosine receptor agonist for A_2A and A3 with K_i of 15 ng/mL and 37 ng/mL, respectively.
M3188	Istradefylline	Istradefylline is a selective adenosine A2A receptor (A2AR) antagonist with K_i of 2.2 nM.
M2282	CGS 21680 hydrochloride	CGS 21680 hydrochloride is an A2A adenosine receptor agonist with an Ki of 27 nM.

Signaling Pathways

Product Type

Adenosine Receptor Adenosine Receptor

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