Adenosine Receptor Adenosine Receptor

Inhibitors

Cat.No.	Name	Information
M4497	Norisoboldine	Norisoboldine is an isoquinoline alkaloid which acts as an AhR agonist.
M7531	AZD4635	AZD4635 is a novel adenosine 2A receptor (A2AR) inhibitor with a Ki of 1.7 nM.
M7282	SCH 58261	SCH 58261 is a potent, highly selective A_2A antagonist.
M2282	CGS 21680 hydrochloride	CGS 21680 hydrochloride is an A2A adenosine receptor agonist with an Ki of 27 nM.
M5211	ZM241385	ZM-241385 is a high affinity antagonist ligand selective for the adenosine A2A receptor.
M20878	Alloxazine	Alloxazine is an A2 receptor antagonist, which is approximately 10-fold more selective for the A2B receptor than for the A2A receptor.
M20848	MIPS521	MIPS521 is a positive allosteric modulator of the A1R that exhibits analgesic efficacy in rats in vivo.
M20627	A2AR antagonist 1	A2AR antagonist 1 is a potent A2AR (Adenosine A2A Receptor) antagonist with Ki values of 4 nM and 264 nM for A2AR and A1R, respectively.
M20421	Theophylline-7-acetic acid	Theophylline-7-acetic acid (Acefylline), acting as an adenosine receptor antagonist, is a stimulant drug of the xanthine chemical class.
M20190	WAY-603264	WAY-603264 is a adenosine kinase inhibitor.
M14295	8-Azaadenosine	8-Azaadenosine is a potent ADAR1 inhibitor and an A-to-I editing inhibitor. 8-Azaadenosine blocks RNA editing and inhibits proliferation, 3D growth, invasion, and migration in thyroid cancer cells.
M13885	5'-N-Ethylcarboxamidoadenosine	5'-N-Ethylcarboxamidoadenosine (NECA) is a nonselective adenosine receptor agonist.
M13884	MRS 1754	MRS 1754 is a selective antagonist radioligand for A_2B adenosine receptor with very low affinity for A₁ and A₃ receptors of both humans and rats.
M13883	LUF6000	LUF6000 is an orally active allosteric modulator of the A3 adenosine receptor. LUF6000 has potent anti-inflammatory effect.
M13882	Adenosine 5'-monophosphate monohydrate	Adenosine 5'-monophosphate monohydrate is an adenosine A₁ receptor agonist. Adenosine 5'-monophosphate monohydrate has significant antiviral activity against HSV-1 and HSV-2.
M11264	KI-7	Ki-7 is an A2B adenosine receptor positive allosteric regulator. Ki-7 enhances cAMP accumulation induced by NECA, a non-selective A2B adenosine receptor agonist (EC50=445.8 nM). Ki-7 also enhanced selective A2B adenosine receptor agonist BAY 60-6583 and adenosine-induced cAMP accumulation with EC50 of 2390 nM and 2550 nM, respectively.
M10628	Adenosine amine congener	Adenosine amine congener (ADAC) is a selective A1 adenosine receptor agonist, can ameliorate noise- and cisplatin-induced cochlear injury.
M10191	Vipadenant	Vipadenant, also known as BIIB014, CEB-4520, is a potent, selective and orally available adenosine A2A receptor antagonist with Ki of 1.3 nM.
M10055	2',5'-Dideoxyadenosine	2′,5′-Dideoxyadenosine is a cell-permeable adenylyl cyclase inhibitor, IC50 = 2.7 μM in detergent-dispersed rat brain preparations.
M9888	ABT-702 dihydrochloride	ABT-702 dihydrochloride is a potent non-nucleoside adenosine kinase inhibitor, selective over other sites of adenosine interaction like A1, A2A and A3 receptors, adenosine transporter and adenosine deaminase.
M9799	Capadenoson	Capadenoson (BAY 68-4986) is an oral active, potent and selective adenosine A1 receptor agonist.
M9774	Namodenoson	Namodenoson (also known as 2-Cl-IB-MECA and CF-102) is an orally bioavailable, synthetic, highly selective adenosine A3 receptor (A3AR) agonist (Ki=0.33 nM) with potential antineoplastic activity.
M9674	MRS-3777 hemioxalate	MRS-3777 hemioxalate is a selective adenosine A3 receptor antagonist.
M9569	Etrumadenant	AB928 is an orally bioavailable, dual antagonist of the A2aR and A2bR adenosine receptors, leads to greater immunomodulatory activity and reduced tumor growth.
M7531	AZD4635	AZD4635 is a novel adenosine 2A receptor (A2AR) inhibitor with a Ki of 1.7 nM.

Signaling Pathways

Product Type

Adenosine Receptor Adenosine Receptor

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