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Adenosine Receptor Adenosine Receptor

Inhibitors

Cat.No.  Name Information
M4497 Norisoboldine Norisoboldine is an isoquinoline alkaloid which acts as an AhR agonist.
M7531 AZD4635 AZD4635 is a novel adenosine 2A receptor (A2AR) inhibitor with a Ki of 1.7 nM.
M7282 SCH 58261 SCH 58261 is a potent, highly selective A2A antagonist.
M2282 CGS 21680 hydrochloride CGS 21680 hydrochloride is an A2A adenosine receptor agonist with an Ki of 27 nM.
M5211 ZM241385 ZM-241385 is a high affinity antagonist ligand selective for the adenosine A2A receptor.
M20878 Alloxazine Alloxazine is an A2 receptor antagonist, which is approximately 10-fold more selective for the A2B receptor than for the A2A receptor.
M20848 MIPS521 MIPS521 is a positive allosteric modulator of the A1R that exhibits analgesic efficacy in rats in vivo.
M20627 A2AR antagonist 1 A2AR antagonist 1 is a potent A2AR (Adenosine A2A Receptor) antagonist with Ki values of 4 nM and 264 nM for A2AR and A1R, respectively.
M20421 Theophylline-7-acetic acid Theophylline-7-acetic acid (Acefylline), acting as an adenosine receptor antagonist, is a stimulant drug of the xanthine chemical class.
M20190 WAY-603264 WAY-603264 is a adenosine kinase inhibitor.
M14295 8-Azaadenosine 8-Azaadenosine is a potent ADAR1 inhibitor and an A-to-I editing inhibitor. 8-Azaadenosine blocks RNA editing and inhibits proliferation, 3D growth, invasion, and migration in thyroid cancer cells.
M13885 5'-N-Ethylcarboxamidoadenosine 5'-N-Ethylcarboxamidoadenosine (NECA) is a nonselective adenosine receptor agonist.
M13884 MRS 1754 MRS 1754 is a selective antagonist radioligand for A2B adenosine receptor with very low affinity for A1 and A3 receptors of both humans and rats.
M13883 LUF6000 LUF6000 is an orally active allosteric modulator of the A3 adenosine receptor. LUF6000 has potent anti-inflammatory effect.
M13882 Adenosine 5'-monophosphate monohydrate Adenosine 5'-monophosphate monohydrate is an adenosine A1 receptor agonist. Adenosine 5'-monophosphate monohydrate has significant antiviral activity against HSV-1 and HSV-2.
M11264 KI-7 Ki-7 is an A2B adenosine receptor positive allosteric regulator. Ki-7 enhances cAMP accumulation induced by NECA, a non-selective A2B adenosine receptor agonist (EC50=445.8 nM). Ki-7 also enhanced selective A2B adenosine receptor agonist BAY 60-6583 and adenosine-induced cAMP accumulation with EC50 of 2390 nM and 2550 nM, respectively.
M10628 Adenosine amine congener Adenosine amine congener (ADAC) is a selective A1 adenosine receptor agonist, can ameliorate noise- and cisplatin-induced cochlear injury.
M10191 Vipadenant Vipadenant, also known as BIIB014, CEB-4520, is a potent, selective and orally available adenosine A2A receptor antagonist with Ki of 1.3 nM.
M10055 2',5'-Dideoxyadenosine 2′,5′-Dideoxyadenosine is a cell-permeable adenylyl cyclase inhibitor, IC50 = 2.7 μM in detergent-dispersed rat brain preparations.
M9888 ABT-702 dihydrochloride ABT-702 dihydrochloride is a potent non-nucleoside adenosine kinase inhibitor, selective over other sites of adenosine interaction like A1, A2A and A3 receptors, adenosine transporter and adenosine deaminase.
M9799 Capadenoson Capadenoson (BAY 68-4986) is an oral active, potent and selective adenosine A1 receptor agonist.
M9774 Namodenoson Namodenoson (also known as 2-Cl-IB-MECA and CF-102) is an orally bioavailable, synthetic, highly selective adenosine A3 receptor (A3AR) agonist (Ki=0.33 nM) with potential antineoplastic activity.
M9674 MRS-3777 hemioxalate MRS-3777 hemioxalate is a selective adenosine A3 receptor antagonist.
M9569 Etrumadenant AB928 is an orally bioavailable, dual antagonist of the A2aR and A2bR adenosine receptors, leads to greater immunomodulatory activity and reduced tumor growth.
M7531 AZD4635 AZD4635 is a novel adenosine 2A receptor (A2AR) inhibitor with a Ki of 1.7 nM.



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