| Cat.No. | Name | Information |
|---|---|---|
| M10191 | Vipadenant | Vipadenant, also known as BIIB014, CEB-4520, is a potent, selective and orally available adenosine A2A receptor antagonist with Ki of 1.3 nM. |
| M10132 | Inosine | Inosine (Inosine) is an endogenous purine nucleoside produced by the catabolism of adenosine. It has immunomodulatory, neuroprotective effects. |
| M7531 | AZD4635 | AZD4635 is a novel adenosine 2A receptor (A2AR) inhibitor with a Ki of 1.7 nM. |
| M7282 | SCH 58261 | SCH 58261 is a potent, highly selective A2A antagonist. |
| M5211 | ZM241385 | ZM-241385 is a high affinity antagonist ligand selective for the adenosine A2A receptor. |
| M4497 | Norisoboldine | Norisoboldine is an isoquinoline alkaloid which acts as an AhR agonist. |
| M3228 | CGS 21680 | CGS 21680 is a selective adenosine receptor agonist for A2A and A3 with Ki of 15 ng/mL and 37 ng/mL, respectively. |
| M2282 | CGS 21680 hydrochloride | CGS 21680 hydrochloride is an A2A adenosine receptor agonist with an Ki of 27 nM. |
| M41758 | DPTN dihydrochloride | DPTN is a potent and selective human, mouse, and rat A3AR antagonist with Ki values of 1.65, 9.61, and 8.53 nM, respectively. |
| M29993 | N6-Cyclohexyladenosine | N6-Cyclohexyladenosine is a selective A1 receptor agonist (EC50 = 8.2 nM). IC50 value: 8.2 nM (EC50) Target: A1 receptor in vivo: N6-Cyclohexyladenosine exerts anticonvulsant effects and protects against neuronal death. CHA was also found to inhibit the pressor effects of lumbar sympathetic nerve stimulation in rats. |
| M20421 | Theophylline-7-acetic acid | Theophylline-7-acetic acid (Acefylline), acting as an adenosine receptor antagonist, is a stimulant agent of the xanthine chemical class. |
| M13885 | 5'-N-Ethylcarboxamidoadenosine | 5'-N-Ethylcarboxamidoadenosine (NECA) is a nonselective adenosine receptor agonist. |
| M13884 | MRS 1754 | MRS 1754 is a selective antagonist radioligand for A2B adenosine receptor with very low affinity for A1 and A3 receptors of both humans and rats. |
| M13882 | Adenosine 5'-monophosphate monohydrate | Adenosine 5'-monophosphate monohydrate is an adenosine A1 receptor agonist. Adenosine 5'-monophosphate monohydrate has significant antiviral activity against HSV-1 and HSV-2. |
| M11264 | KI-7 | Ki-7 is an A2B adenosine receptor positive allosteric regulator. Ki-7 enhances cAMP accumulation induced by NECA, a non-selective A2B adenosine receptor agonist (EC50=445.8 nM). Ki-7 also enhanced selective A2B adenosine receptor agonist BAY 60-6583 and adenosine-induced cAMP accumulation with EC50 of 2390 nM and 2550 nM, respectively. |
| M10628 | Adenosine amine congener | Adenosine amine congener (ADAC) is a selective A1 adenosine receptor agonist, can ameliorate noise- and cisplatin-induced cochlear injury. |
| M9799 | Capadenoson | Capadenoson (BAY 68-4986) is an oral active, potent and selective adenosine A1 receptor agonist. |
| M9774 | Namodenoson | Namodenoson (also known as 2-Cl-IB-MECA and CF-102) is an orally bioavailable, synthetic, highly selective adenosine A3 receptor (A3AR) agonist (Ki=0.33 nM) with potential antineoplastic activity. |
| M9569 | Etrumadenant | Etrumadenant (AB928, A2aR/A2bR antagonist-1) is an orally bioavailable, dual antagonist of the A2aR and A2bR adenosine receptors, leads to greater immunomodulatory activity and reduced tumor growth. |
| M9345 | Preladenant | Preladenant is a potent and competitive antagonist of the human adenosine A2A receptor with a Ki of 1.1 nM. |
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