Inhibitors
Cat.No. | Name | Information |
---|---|---|
M4497 | Norisoboldine | Norisoboldine is an isoquinoline alkaloid which acts as an AhR agonist. |
M7531 | AZD4635 | AZD4635 is a novel adenosine 2A receptor (A2AR) inhibitor with a Ki of 1.7 nM. |
M11264 | KI-7 | Ki-7 is an A2B adenosine receptor positive allosteric regulator. Ki-7 enhances cAMP accumulation induced by NECA, a non-selective A2B adenosine receptor agonist (EC50=445.8 nM). Ki-7 also enhanced selective A2B adenosine receptor agonist BAY 60-6583 and adenosine-induced cAMP accumulation with EC50 of 2390 nM and 2550 nM, respectively. |
M10628 | Adenosine amine congener | Adenosine amine congener (ADAC) is a selective A1 adenosine receptor agonist, can ameliorate noise- and cisplatin-induced cochlear injury. |
M10191 | Vipadenant | Vipadenant, also known as BIIB014, CEB-4520, is a potent, selective and orally available adenosine A2A receptor antagonist with Ki of 1.3 nM. |
M10055 | 2',5'-Dideoxyadenosine | 2′,5′-Dideoxyadenosine is a cell-permeable adenylyl cyclase inhibitor, IC50 = 2.7 μM in detergent-dispersed rat brain preparations. |
M9888 | ABT-702 dihydrochloride | ABT-702 dihydrochloride is a potent non-nucleoside adenosine kinase inhibitor, selective over other sites of adenosine interaction like A1, A2A and A3 receptors, adenosine transporter and adenosine deaminase. |
M9799 | Capadenoson | Capadenoson (BAY 68-4986) is an oral active, potent and selective adenosine A1 receptor agonist. |
M9774 | Namodenoson | Namodenoson (also known as 2-Cl-IB-MECA and CF-102) is an orally bioavailable, synthetic, highly selective adenosine A3 receptor (A3AR) agonist (Ki=0.33 nM) with potential antineoplastic activity. |
M9674 | MRS-3777 hemioxalate | MRS-3777 hemioxalate is a selective adenosine A3 receptor antagonist. |
M9569 | Etrumadenant | AB928 is an orally bioavailable, dual antagonist of the A2aR and A2bR adenosine receptors, leads to greater immunomodulatory activity and reduced tumor growth. |
M7531 | AZD4635 | AZD4635 is a novel adenosine 2A receptor (A2AR) inhibitor with a Ki of 1.7 nM. |
M7282 | SCH 58261 | SCH 58261 is a potent, highly selective A2A antagonist. |
M6126 | CPI-444 | CPI-444 is a potent and selective inhibitor of A2A receptor (A2AR) induces antitumor responses. |
M5924 | Regadenoson | Regadenoson is an A2A adenosine receptor agonist that is a coronary vasodilator that is commonly used in pharmacologic stress testing. |
M5211 | ZM241385 | ZM-241385 is a high affinity antagonist ligand selective for the adenosine A2A receptor. |
M4694 | Theobromine | Theobromine is a methylxanthine found in cocoa beans that inhibits adenosine receptor A1 (AR1) signaling. |
M4497 | Norisoboldine | Norisoboldine is an isoquinoline alkaloid which acts as an AhR agonist. |
M3749 | Pentostatin | Pentostatin (Deoxycoformycin) is an irreversible inhibitor of adenosine deaminase (Ki = 2.5 pM). |
M3228 | CGS 21680 | CGS 21680 is a selective adenosine receptor agonist for A2A and A3 with Ki of 15 ng/mL and 37 ng/mL, respectively. |
M3188 | Istradefylline | Istradefylline is a selective adenosine A2A receptor (A2AR) antagonist with Ki of 2.2 nM. |
M2282 | CGS 21680 hydrochloride | CGS 21680 hydrochloride is an A2A adenosine receptor agonist with an Ki of 27 nM. |
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