| Cat.No. | Name | Information |
|---|---|---|
| M4497 | Norisoboldine | Norisoboldine is an isoquinoline alkaloid which acts as an AhR agonist. |
| M7531 | AZD4635 | AZD4635 is a novel adenosine 2A receptor (A2AR) inhibitor with a Ki of 1.7 nM. |
| M7282 | SCH 58261 | SCH 58261 is a potent, highly selective A2A antagonist. |
| M2282 | CGS 21680 hydrochloride | CGS 21680 hydrochloride is an A2A adenosine receptor agonist with an Ki of 27 nM. |
| M10132 | Inosine | Inosine (Inosine) is an endogenous purine nucleoside produced by the catabolism of adenosine. It has immunomodulatory, neuroprotective effects. |
| M5211 | ZM241385 | ZM-241385 is a high affinity antagonist ligand selective for the adenosine A2A receptor. |
| M3228 | CGS 21680 | CGS 21680 is a selective adenosine receptor agonist for A2A and A3 with Ki of 15 ng/mL and 37 ng/mL, respectively. |
| M10191 | Vipadenant | Vipadenant, also known as BIIB014, CEB-4520, is a potent, selective and orally available adenosine A2A receptor antagonist with Ki of 1.3 nM. |
| M56109 | PD 117519 | PD 117519 (CI947) is an A2A adenosine agonist which has shown oral antihypertensive activity in pharmacological animal models. |
| M56108 | Apadenoson | Apadenoson is an adenosine analog with selective agonist activity for the adenosine A2a receptor and induces coronary vasodilatation. |
| M56107 | Binodenoson | Binodenoson (MRE-0470) is a potent and selective A2A adenosine receptor agonist (KD=270 nM). |
| M56106 | A2B receptor antagonist 2 | A2B receptor antagonist 2 is an adenosine receptor A2B antagonist, with Ki values of 2.30 μM, 6.8 μM and 3.44 μM for rA1, rA2A and hA2B, respectively. |
| M56105 | (±)-5'-Chloro-5'-deoxy-ENBA | (±)-5'-Chloro-5'-deoxy-ENBA is an agonist of A1AR. |
| M56104 | APNEA | APNEA (N6-[2-(4-Aminophenyl)ethyl]adenosine) is a potent, non-selective A3 adenosine receptor agonist. |
| M54826 | LUF5519 | LUF5519 is a ribose-containing adenosine A1 receptor agonist. |
| M54824 | LUF6258 | LUF6258 is a hybrid ortho/allosteric ligand of the adenosine A(1) receptor. |
| M41763 | A3AR agonist 1 | A3AR agonist 1 is an A3AR agonist (Ki: 25.8 nM). |
| M41762 | A3AR agonist 2 | A3AR agonist 2 a selective A3AR agonist (Ki: 22.1 nM). |
| M41761 | Inupadenant hydrochloride | Inupadenant (EOS-850) hydrochloride is an orally active, highly selective A2A receptor antagonist. |
| M41760 | A1/A3 AR antagonist 3 | A1/A3 AR antagonist 3 is an A1R/A3R dual antagonist with high affinity at low-micromolar to low-nanomolar. |
| M41759 | Adenosine receptor antagonist 4 | Adenosine receptor antagonist 4 is an adenosine A1 receptor antagonist with a Ki of 101 nM for human A1 receptor. |
| M41757 | PSB-1901 | PSB-1901 is a potent A2B adenosine receptor (A2BAR) antagonist with Kis of 0.0835 nM and 0.131 nM for human and mouse A2BARs respectively. |
| M41756 | PSB 0777 ammonium hydrate | PSB 0777 ammonium hydrate is a potent and selective adenosine A2A receptor full agonist with Ki values of 44.4 nM, 360 nM for rat and human A2A receptors, respectively. |
| M40667 | A2A receptor antagonist 2 | A2A receptor antagonist 2 is a potent, highly selective adenosine receptor A2A antagonist with an IC50 value of 8.3 nM. |
| M40666 | A2AAR/HDAC-IN-1 | A2AAR/HDAC-IN-1 is an orally active A2AAR/HDAC inhibitor with anticancer activity with a Ki of 163.5 nM for A2AAR and an IC50 of 145.3 nM for HDAC1. |
| M40665 | LJ-4517 | LJ-4517 is a potent adenosine receptor A2AAR antagonist with a Ki of 18.3 nM. |
| M40664 | Adenosine receptor inhibitor 1 | Adenosine receptor inhibitor 1 is a potent, selective adenosine receptor inhibitor with Ki values of >1000, 68.5, >1000, >1000, >1000 nM for A1AR, A2AAR, A2BAR, and A3AR, respectively, and possesses analgesic as well as anti-inflammatory activity. It has analgesic and anti-inflammatory activities and can be used in cancer and neurodegenerative disease research. |
| M40663 | A2A receptor antagonist 3 | A2A receptor antagonist 3 is an adenosine receptor A2a antagonist with a Ki of 0.4 nM. It binds to A2b, A1, and A3 receptors with Ki values of 37, 107, and 1467 nM, respectively. |
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