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Vipadenant, also known as BIIB014, CEB-4520, is a potent, selective and orally available adenosine A2A receptor antagonist with Ki of 1.3 nM. Vipadenant is less potent for A1 with Ki of 69 nM. Vipadenant demonstrates strong oral activity in commonly used models of Parkinson's disease.
Nanyang Technological University. 2024.
Development of smart optical nanoagents for cancer immunotheranostics
Vipadenant purchased from AbMole
| Molecular Weight | 321.34 |
| Formula | C16H15N7O |
| CAS Number | 442908-10-3 |
| Solubility (25°C) | DMSO 30 mg/mL |
| Storage |
Powder -20°C 3 years ; 4°C 2 years In solvent -80°C 6 months ; -20°C 1 month |
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| FK 453
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| GS-9667
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| PD81723
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| PSB-0788
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Products are for research use only. Not for human use. We do not sell to patients.
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