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SCH 58261 is a potent and selective A2A adenosine receptor competitive antagonist (Ki = 1.3 nM). SCH 58261 displays 323-, 53- and 100-fold selectivity over A1, A2B and A3 receptors, respectively.
Front Pharmacol. 2022 Jun 23;13:897436.
Xiaoyaosan Ameliorates Chronic Restraint Stress-Induced Depression-Like Phenotype by Suppressing A2AR Signaling in the Rat Striatum
SCH 58261 purchased from AbMole
| Molecular Weight | 345.36 |
| Formula | C18H15N7O |
| CAS Number | 160098-96-4 |
| Solubility (25°C) | DMSO 30 mg/mL |
| Storage |
Powder -20°C 3 years ; 4°C 2 years In solvent -80°C 6 months ; -20°C 1 month |
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