| Cat.No. | Name | Information |
|---|---|---|
| M4497 | Norisoboldine | Norisoboldine is an isoquinoline alkaloid which acts as an AhR agonist. |
| M7531 | AZD4635 | AZD4635 is a novel adenosine 2A receptor (A2AR) inhibitor with a Ki of 1.7 nM. |
| M7282 | SCH 58261 | SCH 58261 is a potent, highly selective A2A antagonist. |
| M2282 | CGS 21680 hydrochloride | CGS 21680 hydrochloride is an A2A adenosine receptor agonist with an Ki of 27 nM. |
| M10132 | Inosine | Inosine (Inosine) is an endogenous purine nucleoside produced by the catabolism of adenosine. It has immunomodulatory, neuroprotective effects. |
| M5211 | ZM241385 | ZM-241385 is a high affinity antagonist ligand selective for the adenosine A2A receptor. |
| M3228 | CGS 21680 | CGS 21680 is a selective adenosine receptor agonist for A2A and A3 with Ki of 15 ng/mL and 37 ng/mL, respectively. |
| M10191 | Vipadenant | Vipadenant, also known as BIIB014, CEB-4520, is a potent, selective and orally available adenosine A2A receptor antagonist with Ki of 1.3 nM. |
| M8825 | Adenosine A1 receptor activator T62 | Adenosine A1 receptor activator T62 is an allosteric enhancer of adenosine A1 receptor. |
| M8751 | BAY 60-6583 | BAY 60-6583 is a potent and high-affinity agonist of adenosine A2B receptor with EC50 of 3 nM. |
| M7713 | 2-Chloroadenosine | 2-Chloroadenosine is a selective A1 adenosine receptor agonist. 2-Chloroadenosine is an apparent competitive inhibitor of uridine influx (apparent Ki=33 μM) and high-affinity nitrobenzylthioinosine binding (apparent Ki=0.18 mM). |
| M7699 | CGS-15943 | Highly potent, non-selective adenosine receptor antagonist. |
| M7307 | SLV 320 | SLV 320 is a potent and selective A 1 antagonist. |
| M7281 | SCH 442416 | SCH 442416 is a very selective, high affinity A 2A antagonist. |
| M7170 | PSB-603 | PSB 603 is a highly selective A 2B antagonist. |
| M6999 | MRS 1706 | MRS 1706 is a potent and selective A 2B inverse agonist. |
| M6803 | Piclidenoson (IB-MECa) | Piclidenoson is a first-in-class and selective A3AR agonist. In vitro, in OVCAR-3 cells, Piclidenoson is able to inhibit forskolin-stimulated cAMP levels with an EC 50 of 0.82 μM. |
| M6689 | DPCPX | DPCPX is a potent and selective A1 adenosine receptor antagonist, both in vitro and in vivo. Ki values are 3.9, 130, 50 and 4000 nM for human A1, A2A, A2B and A3 receptors respectively. |
| M6359 | 8-Cyclopentyl-1,3-dimethylxanthine | 8-Cyclopentyl-1,3-dimethylxanthine is a high affinity adenosine A 1 receptor antagonist. |
| M6357 | 8-Aminoadenine | 8-Aminoadenine is a adenine receptor agonist. |
| M6126 | CPI-444 | CPI-444 is a potent and selective inhibitor of A2A receptor (A2AR) induces antitumor responses. |
| M5924 | Regadenoson | Regadenoson is an A2A adenosine receptor agonist that is a coronary vasodilator that is commonly used in pharmacologic stress testing. |
| M5057 | Proxyphylline | Proxyphylline is a methylxanthine and derivative of theophylline. |
| M4694 | Theobromine | Theobromine is a methylxanthine found in cocoa beans that inhibits adenosine receptor A1 (AR1) signaling. |
| M3188 | Istradefylline | Istradefylline (KW-6002) is a potent, selective and orally active adenosine A2A receptor (A2AR) antagonist with Ki of 2.2 nM. |
| M1864 | SYN115 | SYN115 is a novel, selective adenosine A(2A) receptor antagonist. |
| M56114 | CV1808 | CV1808 (2-Phenylaminoadenosine) is a non-selective A2 adenosine receptor (A2 AR) agonist with Kis of 76 and 1450 nM for A2A and A3 adenosine receptor subtypes, respectively. |
| M56113 | FK 453 | FK 453 is a potent and selective adenosine A1 receptor antagonist with an IC50 value of 17.2 nM. |
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