| Cat.No. | Name | Information |
|---|---|---|
| M4497 | Norisoboldine | Norisoboldine is an isoquinoline alkaloid which acts as an AhR agonist. |
| M7531 | AZD4635 | AZD4635 is a novel adenosine 2A receptor (A2AR) inhibitor with a Ki of 1.7 nM. |
| M7282 | SCH 58261 | SCH 58261 is a potent, highly selective A2A antagonist. |
| M2282 | CGS 21680 hydrochloride | CGS 21680 hydrochloride is an A2A adenosine receptor agonist with an Ki of 27 nM. |
| M10132 | Inosine | Inosine (Inosine) is an endogenous purine nucleoside produced by the catabolism of adenosine. It has immunomodulatory, neuroprotective effects. |
| M5211 | ZM241385 | ZM-241385 is a high affinity antagonist ligand selective for the adenosine A2A receptor. |
| M3228 | CGS 21680 | CGS 21680 is a selective adenosine receptor agonist for A2A and A3 with Ki of 15 ng/mL and 37 ng/mL, respectively. |
| M10191 | Vipadenant | Vipadenant, also known as BIIB014, CEB-4520, is a potent, selective and orally available adenosine A2A receptor antagonist with Ki of 1.3 nM. |
| M7713 | 2-Chloroadenosine | 2-Chloroadenosine is a selective A1 adenosine receptor agonist. 2-Chloroadenosine is an apparent competitive inhibitor of uridine influx (apparent Ki=33 μM) and high-affinity nitrobenzylthioinosine binding (apparent Ki=0.18 mM). |
| M7699 | CGS-15943 | Highly potent, non-selective adenosine receptor antagonist. |
| M7307 | SLV 320 | SLV 320 is a potent and selective A 1 antagonist. |
| M7281 | SCH 442416 | SCH 442416 is a very selective, high affinity A 2A antagonist. |
| M7170 | PSB-603 | PSB 603 is a highly selective A 2B antagonist. |
| M6999 | MRS 1706 | MRS 1706 is a potent and selective A 2B inverse agonist. |
| M6803 | Piclidenoson (IB-MECa) | Piclidenoson is a first-in-class and selective A3AR agonist. In vitro, in OVCAR-3 cells, Piclidenoson is able to inhibit forskolin-stimulated cAMP levels with an EC 50 of 0.82 μM. |
| M6359 | 8-Cyclopentyl-1,3-dimethylxanthine | 8-Cyclopentyl-1,3-dimethylxanthine is a high affinity adenosine A 1 receptor antagonist. |
| M6357 | 8-Aminoadenine | 8-Aminoadenine is a adenine receptor agonist. |
| M6126 | CPI-444 | CPI-444 is a potent and selective inhibitor of A2A receptor (A2AR) induces antitumor responses. |
| M5924 | Regadenoson | Regadenoson is an A2A adenosine receptor agonist that is a coronary vasodilator that is commonly used in pharmacologic stress testing. |
| M5057 | Proxyphylline | Proxyphylline is a methylxanthine and derivative of theophylline. |
| M4694 | Theobromine | Theobromine is a methylxanthine found in cocoa beans that inhibits adenosine receptor A1 (AR1) signaling. |
| M3188 | Istradefylline | Istradefylline (KW-6002) is a potent, selective and orally active adenosine A2A receptor (A2AR) antagonist with Ki of 2.2 nM. |
| M1864 | SYN115 | SYN115 is a novel, selective adenosine A(2A) receptor antagonist. |
| M56114 | CV1808 | CV1808 (2-Phenylaminoadenosine) is a non-selective A2 adenosine receptor (A2 AR) agonist with Kis of 76 and 1450 nM for A2A and A3 adenosine receptor subtypes, respectively. |
| M56113 | FK 453 | FK 453 is a potent and selective adenosine A1 receptor antagonist with an IC50 value of 17.2 nM. |
| M56112 | GS-9667 | GS-9667 (CVT 3619), a novel N6-5'-substituted adenosine analog, is a selective, partial agonist of the A1 adenosine receptor (A1AdoR). |
| M56111 | PD81723 | PD81723 is an adenosine receptor binding enhancer. |
| M56110 | PSB-0788 | PSB-0788 is a new selective high-affinity A2B antagonist with IC50 value of 3.64 nM and Ki value of 0.393 nM, respeactively. |
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