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Piclidenoson (IB-MECa)

Cat. No. M6803

All AbMole products are for research use only, cannot be used for human consumption.

Piclidenoson (IB-MECa) Structure
Synonym:

CF-101

Size Price Availability Quantity
2mg USD 40  USD40 In stock
5mg USD 70  USD70 In stock
10mg USD 110  USD110 In stock
25mg USD 235  USD235 In stock
50mg USD 370  USD370 In stock
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Quality Control & Documentation
Biological Activity

Piclidenoson is a first-in-class and selective A3AR agonist.  In vitro, in OVCAR-3 cells, Piclidenoson is able to inhibit forskolin-stimulated cAMP levels with an EC 50 of 0.82 μM.

Chemical Information
Molecular Weight 510.29
Formula C18H19IN6O4
CAS Number 152918-18-8
Form Solid
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Lashinger, et al. Am J Physiol Renal Physiol. AMTB, a TRPM8 channel blocker: evidence in rats for activity in overactive bladder and painful bladder syndrome.

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  Catalog
Abmole Inhibitor Catalog




Keywords: Piclidenoson (IB-MECa), CF-101 supplier, Adenosine Receptor, inhibitors, activators

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