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 About 30 results found for searched term "Opioid Receptor" (0.019 seconds)

Cat.No.  Name Information
M1953 ADL5859 Hydrochloride ADL5859 is a potent, selective and orally bioavailable δ-opioid receptor agonist (Ki = 0.84 nM, EC50 = 20 nM).
M2145 Loperamide hydrochloride Loperamide hydrochloride is a high affinity μ-opioid receptor agonist with peripheral selectivity with Ki values of 2, 48 and 1156 nM for μ-, δ- and κ-opioid receptors respectively. Loperamide hydrochloride is also a selective and competitive human intestinal carboxylesterases (hiCE) inhibitor.
M2214 JTC-801 JTC-801 is a novel opioid receptor-like1 (ORL1) receptor antagonist with IC50 of 94 nM.
M2875 Nalmefene hydrochloride Nalmefene is an opioid receptor antagonist, it is used primarily in the management of alcohol dependence.
M2991 SA 4503 dihydrochloride SA 4503 is a novel and selective opioid sigma1 receptor agonist with IC50 of 17.4 nM.
M1577 Naltrexone Hydrochloride Naltrexone hydrochlorideis an opioid receptor antagonist used primarily in the management of alcohol dependence and opioid dependence.
M4456 Sec-O-Glucosylhamaudol Sec-o-glucosylhamaudol is a natural product isolated from The apostrophophore, which can reduce the protein level of μ-opioid receptor and can be used for pain relief research.
M4516 Sinomenine-Hydrochloride Sinomenine hydrochloride (Cucoline hydrochloride), an alkaloid derived from Sinomenium Acutum, is a blocker of NF-κB activation. Sinomenine is also a μ-opioid receptor activator.
M4520 (+)-Corydaline Corydaline ((+) -corydaline) is an isoquinoline alkaloid extracted from Corydalis Yanhusuo. It is an inhibitor of AChE with IC50 of 226 µM. Corydaline is a μ-opioid receptor agonist (Ki = 1.23 µM) that inhibits the replication of enterovirus 71 (EV71) (IC50 = 25.23 µM). Corydaline has anti-angiogenesis, anti-allergy, gastric emptying and anti-nociception effects.
M4808 TRV130 hydrochloride TRV130 (Oliceridine) hydrochloride is a novel μ-opioid receptor (MOR) G protein-biased ligand.
M5065 Cebranopadol Cebranopadol is a NOP and opioid receptor agonist that acts on human NOP, MOP, KOP and δ-opioid peptide (DOP) receptors with Ki/EC50 values of 0.9 nM/13 nM and 0.7 nM/1.2 nM, respectively. 2.6 nM/17 nM, 18 nM/110 nM.
M5067 Eluxadoline Eluxadoline is an orally active mixed μ opioid receptor (μOR) agonist δ opioid receptor (δOR) antagonist.
M5289 PZM21 PZM21 is a potent and selective μ-opioid-receptor (μOR) agonist with an EC50 of 1.8 nM.
M5403 Alvimopan dihydrate Alvimopan dihydrate (ADL 8-2698 dihydrate) is a potent, selective, orally active and reversible μ-opioid receptor antagonist, with an IC50 of 1.7 nM. Alvimopan dihydrate has selectivity for μ-opioid receptor (Ki=0.47 nM) over κ- and δ-opioid receptors (Kis=100, 12 nM, respectively).
M7882 Levallorphan tartrate salt Partial agonist (antagonist) at μ and δ opioid receptors.
M7946 Naloxone methiodide Quaternary salt of naloxone that, like the parent compound, is a nonselective antagonist at opioid receptors.
M7951 Naltrindole isothiocyanate hydrochloride Naltrindole isothiocyanate hydrochloride is a selective irreversible δ2 opioid receptor antagonist.
M7984 Opipramol dihydrochloride σ12 opioid receptor agonist; an antagonist at D2, 5HT2 and H1 receptors; atypical antidepressant, antipsychotic and anxiolytic.
M8030 PB28 dihydrochloride Selective σ2 opioid receptor ligand; putative σ2 agonist.
M8191 Salvinorin A Salvinorin A is a potent, non-nitrogenous κ opioid selective receptor agonist.
M8453 ML138 ML138 (CID 44601470) is a highly selective agonist at kappa opioid receptors (KOR) that potently activate G protein coupling but weakly interact with β arrestin2.
M8502 Alvimopan Alvimopan is a gastroprokinetic peripheral mu-opioid receptor antagonist.
M8776 ARM390 ARM390 in a δ-selective opioid receptor agonist derivative of SNC80.
M8832 U-69593 U-69593 is a selective κ opioid receptor agonist.
M8834 U-62066 Highly selective κ opioid receptor agonist; antitussive.
M9268 Met-Enkephalin Met-Enkephalin (H-Tyr-Gly-Gly-Phe-Met-OH) inhibits tumor growth via binding to the opioid receptor.
M9514 JDTic JDTic is a kappa opioid receptor (KOR) antagonist that prevents stress-induced reinstatement of cocaine-maintained responding and has antidepressant-like effects.
M9615 DAMGO DAMGO is an opioid receptor agonist with the ability to affect the locomotive activity in rodents, Kd value is 3.46 nM for native μ-OPR.
M10229 Porcine dynorphin A (1-13) Porcine dynorphin A (1-13) is a potent, endogenous κ opioid receptor agonist.
M10240 CTOP TFA CTOP TFA is a peptide that acts as a potent and selective μ opioid receptor antagonist, with Ki values of 0.96 and >10,000 nM for μ and δ receptors, respectively.

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