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 About 30 results found for searched term "Opioid Receptor" (0.051 seconds)

Cat.No.  Name Target
M1953 ADL5859 Hydrochloride Opioid Receptor
ADL5859 HCl
ADL5859 is a potent, selective and orally bioavailable δ-opioid receptor agonist (Ki = 0.84 nM, EC50 = 20 nM).
M2145 Loperamide hydrochloride Animal Modeling
R-18553 hydrochloride
Loperamide hydrochloride is a high affinity μ-opioid receptor agonist with peripheral selectivity with Ki values of 2, 48 and 1156 nM for μ-, δ- and κ-opioid receptors respectively. Loperamide hydrochloride is also a selective and competitive human intestinal carboxylesterases (hiCE) inhibitor. It can be used to construct animal models of functional constipation.
M2214 JTC-801 Opioid Receptor
JTC-801 is a novel opioid receptor-like1 (ORL1) receptor antagonist with IC50 of 94 nM.
M2875 Nalmefene hydrochloride Opioid Receptor
Nalmefene is an opioid receptor antagonist, it is used primarily in the management of alcohol dependence.
M2991 SA 4503 dihydrochloride Opioid Receptor
AGY94806 dihydrochloride; Cutamesine dihydrochloride
SA 4503 is a novel and selective opioid sigma1 receptor agonist with IC50 of 17.4 nM.
M1577 Naltrexone Hydrochloride Opioid Receptor
Naltrexone hydrochlorideis an opioid receptor antagonist used primarily in the management of alcohol dependence and opioid dependence.
M4456 Sec-O-Glucosylhamaudol Opioid Receptor
Sec-o-glucosylhamaudol is a natural product isolated from The apostrophophore, which can reduce the protein level of μ-opioid receptor and can be used for pain relief research.
M4516 Sinomenine-Hydrochloride NF-κB
Cucoline hydrochloride
Sinomenine hydrochloride (Cucoline hydrochloride), an alkaloid derived from Sinomenium Acutum, is a blocker of NF-κB activation. Sinomenine is also a μ-opioid receptor activator.
M4520 (+)-Corydaline AChR/AChE
(+)-Corydaline; Corydalin
Corydaline ((+) -corydaline) is an isoquinoline alkaloid extracted from Corydalis Yanhusuo. It is an inhibitor of AChE with IC50 of 226 µM. Corydaline is a μ-opioid receptor agonist (Ki = 1.23 µM) that inhibits the replication of enterovirus 71 (EV71) (IC50 = 25.23 µM). Corydaline has anti-angiogenesis, anti-allergy, gastric emptying and anti-nociception effects.
M4808 TRV130 hydrochloride Opioid Receptor
Oliceridine HCl; TRV130 HCl
TRV130 (Oliceridine) hydrochloride is a novel μ-opioid receptor (MOR) G protein-biased ligand.
M5065 Cebranopadol Opioid Receptor
Cebranopadol is a NOP and opioid receptor agonist that acts on human NOP, MOP, KOP and δ-opioid peptide (DOP) receptors with Ki/EC50 values of 0.9 nM/13 nM and 0.7 nM/1.2 nM, respectively. 2.6 nM/17 nM, 18 nM/110 nM.
M5067 Eluxadoline Opioid Receptor
Eluxadoline is an orally active mixed μ opioid receptor (μOR) agonist δ opioid receptor (δOR) antagonist.
M5289 PZM21 Opioid Receptor
PZM21 is a potent and selective μ-opioid-receptor (μOR) agonist with an EC50 of 1.8 nM.
M5403 Alvimopan dihydrate Opioid Receptor
LY 246736 dihydrate; ADL 8-2698 dihydrate
Alvimopan dihydrate (ADL 8-2698 dihydrate) is a potent, selective, orally active and reversible μ-opioid receptor antagonist, with an IC50 of 1.7 nM. Alvimopan dihydrate has selectivity for μ-opioid receptor (Ki=0.47 nM) over κ- and δ-opioid receptors (Kis=100, 12 nM, respectively).
M7882 Levallorphan tartrate salt Others
Partial agonist (antagonist) at μ and δ opioid receptors.
M7946 Naloxone methiodide Others
Quaternary salt of naloxone that, like the parent compound, is a nonselective antagonist at opioid receptors.
M7951 Naltrindole isothiocyanate hydrochloride Others
Naltrindole isothiocyanate hydrochloride is a selective irreversible δ2 opioid receptor antagonist.
M7984 Opipramol dihydrochloride Others
σ12 opioid receptor agonist; an antagonist at D2, 5HT2 and H1 receptors; atypical antidepressant, antipsychotic and anxiolytic.
M8030 PB28 dihydrochloride Others
Selective σ2 opioid receptor ligand; putative σ2 agonist.
M8191 Salvinorin A Others
Salvinorin A is a potent, non-nitrogenous κ opioid selective receptor agonist.
M8453 ML138 Others
ML138 (CID 44601470) is a highly selective agonist at kappa opioid receptors (KOR) that potently activate G protein coupling but weakly interact with β arrestin2.
M8502 Alvimopan Opioid Receptor
ADL 8-2698; LY 246736
Alvimopan is a gastroprokinetic peripheral mu-opioid receptor antagonist.
M8776 ARM390 Others
ARM390 in a δ-selective opioid receptor agonist derivative of SNC80.
M8832 U-69593 Opioid Receptor
U-69593 is a selective κ opioid receptor agonist.
M8834 U-62066 Others
Highly selective κ opioid receptor agonist; antitussive.
M9268 Met-Enkephalin Opioid Receptor
Met-Enkephalin (H-Tyr-Gly-Gly-Phe-Met-OH) inhibits tumor growth via binding to the opioid receptor.
M9514 JDTic Opioid Receptor
JDTic is a kappa opioid receptor (KOR) antagonist that prevents stress-induced reinstatement of cocaine-maintained responding and has antidepressant-like effects.
M9615 DAMGO Opioid Receptor
RX783006; Dagol
DAMGO is an opioid receptor agonist with the ability to affect the locomotive activity in rodents, Kd value is 3.46 nM for native μ-OPR.
M10229 Porcine dynorphin A (1-13) Opioid Receptor
Dynorphin A Porcine Fragment 1-13
Porcine dynorphin A (1-13) is a potent, endogenous κ opioid receptor agonist.
M10240 CTOP TFA Opioid Receptor
CTOP TFA is a peptide that acts as a potent and selective μ opioid receptor antagonist, with Ki values of 0.96 and >10,000 nM for μ and δ receptors, respectively.

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