About 32 results found for searched term "ATPA" (0.107 seconds)
| Cat.No. | Name | Target |
|---|---|---|
| M7593 | ATPA | Others |
| Selective kainate receptor agonist. | ||
| M56515 | ATPA | GluR |
| ATPA is a selective glutamate receptor GluR5 activator with EC50s of 0.66, 9.5, 1.4, 23, 32, 18, and 14 μM for GluR5wt, GluR5(S741M), GluR5(S721T), GluR5(S721T, S741M), GluR5(S741A), GluR5(S741L), and GluR5(S741V), respectively. | ||
| M2093 | Enoxacin | Anti-infection |
| AT 2266; CI 919 | ||
| Enoxacin is a small molecule inhibitor of binding between the B2-subunit of vacuolar H+-ATPase (V-ATPase) and microfilaments. | ||
| M2294 | Brefeldin A | ATPase |
| BFA; Cyanein; Decumbin | ||
| Brefeldin A is a lactone antibiotic and ATPase inhibitor for protein transport with IC50 of 0.2 μM in HCT 116 cells. Brefeldin A is also an autophagy and mitophagy inhibitor. Brefeldin A is a CRISPR/Cas9 activator. Brefeldin A inhibits HSV-1 and has anti-cancer activity. | ||
| M2459 | (-)-Blebbistatin | Myosin |
| (S)-(-)-Blebbistatin | ||
| (-)-Blebbistatin is a cell-permeable inhibitor for non muscle myosin II ATPase with IC50 of ~2 μM, does not inhibit myosin light chain kinase, inhibits contraction of the cleavage furrow without disrupting mitosis or contractile ring assembly. *The compound is unstable in solutions, freshly prepared is recommended | ||
| M2474 | BTB06584 | ATPase |
| BTB06584 is an IF1-dependent, selective inhibitor of the mitochondrial F1 Fo-ATPase. | ||
| M3449 | PF-3716556 | Potassium Channel |
| PF 3716556 is a potent and selective P-CAB (potassium-competitive acid blocker), with pIC50 of 6.026 and 7.095 for the inhibition of porcine H+,K+-ATPase activity in ion-leaky and ion-tight assay, respectively, inhibits gastric acid secretion, displays no activity at Na+ | ||
| M3696 | Rostafuroxin | ATPase |
| PST 2238 | ||
| Rostafuroxin, a novel antihypertensive compound, acts as a selective inhibitor of srC-SH2 interaction with Na, K-ATPase activated by mutated adducin and Wabin in vivo. | ||
| M3707 | Rabeprazole Sodium | Proton Pump |
| LY307640 sodium | ||
| Rabeprazole is a frequently used second-generation proton pump inhibitor (PPI) that irreversibly inactivates gastric H+/K+-ATPase. | ||
| M3987 | Ginsenoside Rb1 | Sodium Channel |
| Gynosaponin C; Gypenoside III | ||
| Ginsenoside Rb1 is an ingredient in the Chinese medicine Panax ginseng. Ginsenoside inhibition Na, K-ATPase++ activityIC50 6.3±1.0 μM. Ginsenoside Rb1 also inhibits IRAK-1 activation and phosphorylation of NF-κB p65. | ||
| M4339 | Bufalin | Sodium Channel |
| Bufalin is a potent Na+/K+-ATPase inhibitor, binds to the subunit α1, α2 and α3, with Kd of 42.5, 45 and 40 nM respectively, it has anti-cancer activity. | ||
| M4606 | Phloridzin | SGLT |
| Floridzin; NSC 2833 | ||
| Phloridzin is a non-selective SGLT inhibitor with Kis of 300 and 39 nM for hSGLT1 and hSGLT2, respectively. Phlorizin is also a Na+/K+-ATPase inhibitor. | ||
| M4765 | Oleandrin | Sodium Channel |
| Oleandrin (PBI-05204) inhibited Na+, K+ -atPase activity with IC50 of 620 nM. | ||
| M4953 | Bafilomycin A1 | Proton Pump |
| Baf-A1；BafA1 | ||
| Bafilomycin A1 (BafA1) is a vacuolar H+-ATPase inhibitor with IC50 of 0.44 nM. | ||
| M5161 | Sodium orthovanadate | ATPase |
| Sodium vanadate | ||
| Sodium orthovanadate is an alkaline phosphatase and (Na,K)-ATPase inhibitor with IC50 of 10 μM. | ||
| M5285 | Ilaprazole | Proton Pump |
| IY-81149 | ||
| Ilaprazole, a substituted benzimidazole, is a new candidate drug that is an H+ /K+ ATPase inhibitor designed for the treatment of gastric ulcers. | ||
| M5409 | Amiodarone hydrochloride | Potassium Channel |
| Amiodarone HCl is a sodium/potassium-ATPase inhibitor and an autophagy activator, used to treat various types of cardiac dysrhythmias. | ||
| M5633 | Pantoprazole sodium | Proton Pump |
| SKF96022 sodium, BY-1023 sodium | ||
| Pantoprazole is a proton pump inhibitor drug that inhibits gastric acid secretion. It works on gastric parietal cells to irreversibly inhibit (H+/K+)-ATPase function and suppress the production of gastric acid. | ||
| M9118 | Chebulinic acid | DNA/RNA Synthesis |
| NSC69862 | ||
| Chebulinic acid is a potent natural inhibitor of M. tuberculosis DNA gyrase, also can inhibit SMAD-3 phosphorylation, inhibit H+ K+-ATPase activity. | ||
| M6194 | Esomeprazole Magnesium trihydrate | Autophagy |
| (S)-Omeprazole magnesium trihydrate | ||
| Esomeprazole Magnesium trihydrate is a proton pump inhibitor which reduces acid secretion through inhibition of the H+ / K+ ATPase in gastric parietal cells. | ||
| M6501 | BHQ | Others |
| 2,5-Di-tert-butylhydroquinone | ||
| BHQ is a inhibitor of SERCA ATPase. | ||
| M6551 | Bz 423 | Others |
| BZ48 | ||
| Bz 423 is a aTP synthase inhibitor (IC50 ~5 μM). Bz 423 binds the oligomycin sensitivity conferring protein (OSCP) component of mitochondrial F1F0-ATPase in vitro resulting in generation of superoxide and apoptosis. Bz 423 kills primary B and T cell in mice in vivo. Bz 423 suppresses autoimmunity and prolongs survival in mouse lupus model. | ||
| M6973 | ML 240 | Others |
| ML 240 is a aTP-competitive inhibitor of p97 ATPase. | ||
| M7103 | Paxilline | Potassium Channel |
| Paxilline is a sERCA ATPase blocker. Also potent BKCa channel blocker. | ||
| M7280 | SCH 28080 | Others |
| SCH 28080 is a h +,K +-ATPase inhibitor. | ||
| M7353 | Tamoxifen | Estrogen Receptor |
| ICI47699; Z-Tamoxifen; trans-Tamoxifen | ||
| Tamoxifen is an orally active, selective estrogen receptor partial agonist/antagonist. Tamoxifen is a potent Hsp90 activator and enhances the Hsp90 molecular chaperone ATPase activity. Tamoxifen also potent inhibits infectious EBOV Zaire and Marburg (MARV) with IC50 of 0.1 µM and 1.8 µM, respectively. | ||
| M7409 | Thapsigargin | Calcium Channel |
| Thapsigargin is an endoplasmic reticulum (ER) stress inducer, it is also an inhibitor of microsomal Ca2+-ATPase. | ||
| M7575 | Apoptozole | HSP |
| Apoptozole is an inhibitor of the ATPase domain of Hsc70 and Hsp70, with Kds of 0.21 and 0.14 μM, respectively, and can induce apoptosis. | ||
| M7624 | 2,3-Butanedione monoxime | Myosin |
| Biacetyl monoxime; Diacetyl monoxime; DAM | ||
| 2,3-Butanedione Monoxime (BDM) is a myosin ATPASE inhibitor. 2,3-Butanedione Monoxime is a skeletal and cardiac muscle contraction inhibitor. 2,3-Butanedione monoxime induces sarcoplasmic reticulum Ca2+ release. | ||
| M7732 | CGP-37157 | Sodium Channel |
| CGP37157 is a potent, selective inhibitor of mitochondrial Na+/Ca2+ exchange as well as sarcoplasmic reticulum calcium-stimulated ATPase and possibly other calcium channels. | ||
| M7737 | Concanamycin A (Folimycin) | ATPase |
| X 4357B; Folimycin; CMA | ||
| Concanamycin A (Folimycin) is a macrolide antibiotic and a specific vacuolar type H+-ATPase (V-ATPase) inhibitor. | ||
| M8185 | Strophanthidin | Others |
| Strophanthidin is a cardiotonic steroid that elevates the activity of Na+/K+-ATPase in cardiac myocytes. | ||
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