Cat.No. | Name | Information |
---|---|---|
M2030 | Apremilast | Apremilast is a novel, orally available small molecule inhibitor of PDE4 with IC50 of 74 nM. |
M6804 | IBMX | IBMX is a pDE inhibitor (non-selective) with IC50 values of 6.5±1.2, 26.3±3.9 and 31.7±5.3 μM for PDE3, 4 and 5 respectively. |
M1906 | Piclamilast | Piclamilast (RP 73401) is a potent and selective inhibitor of phosphodiesterase (PDE) 4. |
M1871 | Roflumilast | Roflumilast (trade names Daxas, Daliresp) is a novel and selective, long-acting inhibitor of phosphodiesterase 4 (PDE-4). |
M1734 | BAY-60-7550 | BAY-60-7550 is a potent PDE2 inhibitor with IC50 values of 2.0 nM (bovine) and 4.7 nM (human). |
M1728 | GSK256066 | GSK256066 is a selective phosphodiesterase 4 (PDE4)inhibitor with an IC50 of 3.2 pM. *The compound is unstable in solutions, freshly prepared is recommended |
M49421 | ME-3183 | ME-3183 is an oral selective PDE4 inhibitor with anti-inflammatory activity for studies related to plaque psoriasis. |
M49420 | ART-648 | ART-648 is a PDE4 inhibitor that may be used in studies related to non-alcoholic steatohepatitis. |
M49402 | (E/Z)-HA155 | (E/Z)-HA155 is a potent Autotaxin (ATX) type I inhibitor for studies related to cancer, fibrous disorders, inflammation, pain and angiogenesis. |
M49401 | Autotaxin-IN-3 | Autotaxin-IN-3 is an Autotaxin(ATX) inhibitor with an IC50 value of 2.4 nM. |
M49400 | HA155 | HA155 is a potent and selective ATX inhibitor with an IC50 value of 5.7 nM. |
M49398 | ATX inhibitor 5 | ATX inhibitor 5 is a potent, orally active inhibitor of Autotaxin (ATX) with an IC50 of 15.3 nM.Additionally, AATX inhibitor 5 exhibits anti-hepatic fibrosis activity and significantly reduces CCl4-induced hepatic fibrosis. |
M49394 | BBT-877 | BBT-877 is an oral small molecule autotaxin (ATX) inhibitor for use in studies related to non-alcoholic steatohepatitis (NASH) and idiopathic pulmonary fibrosis (IPF). |
M44885 | Ilexsaponin B2 | Ilexsaponin B2 is a saponin isolated from the root of Ilex pubescens Hook. |
M42569 | Enpp-1-IN-16 | Enpp-1-IN-16 is an ENPP1 inhibitor. |
M42568 | cis-Tadalafil | cis-Tadalafil is a PDE5 inhibitor (IC50: 0.09 μM). |
M42567 | Motapizone | Motapizone (NAT 05-239) is a selective PDE3 inhibitor. |
M42566 | PDE4-IN-13 | PDE4-IN-13 is a PDE4 inhibitor with an IC50 of 1.56 μM. |
M42565 | PDE1-IN-5 | PDE1-IN-5 is a selective PDE1C inhibitor (IC50: 15 nM). |
M42564 | CD00509 | CD00509 is a Tdp1 inhibitor, with an IC50 value of 0.71 μM. |
M42563 | PDE5-IN-10 | PDE5-IN-10 is a potent PDE5 inhibitor with an IC50 of 20 nM. |
M42562 | ATX inhibitor 18 | ATX inhibitor 18 is a potent ATX inhibitor with an IC50 value of 24.2 nM. |
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